Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 2 of 2: Calculated dose response metrics. - Dataset (ID:20351)
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Cell | Small Molecule | Treatment Duration | GR50 | GRmax | GR_AOC | GEC50 | GRinf | hGR |
---|---|---|---|---|---|---|---|---|
CAMA-1 | SB1-F-22 | 72 | 43.6088606735 | 0.4408 | 0.0565 | 156.5267 | -1.0000 | 0.8597 |
HCC1428 | z-VAE(OMe)-fmk | 72 | inf | 0.9944 | 0.0566 | 0.0000 | 0.9577 | 0.0100 |
PDXHCI002 | z-VAE(OMe)-fmk | 72 | inf | 0.9278 | 0.0585 | 0.0000 | 0.9445 | 0.0100 |
SK-BR-3 | USP7-IN-1 | 72 | 62.2210904101 | 0.5764 | 0.0588 | 133.0943 | -1.0000 | 1.4449 |
MDA-MB-134-VI | HY-17542 | 72 | inf | 0.5701 | 0.0598 | 0.0000 | 0.9013 | 0.0100 |
MDA-MB-231 | IU1 | 72 | inf | 0.8503 | 0.0614 | 0.0000 | 0.9320 | 0.0100 |
T47D | SB1-F-22 | 72 | 156.804339896 | 0.7134 | 0.0621 | 286.2396 | -0.2481 | 0.6696 |
MDA-MB-134-VI | ML-323 | 72 | 45.5586104943 | 0.3266 | 0.0626 | 58.1271 | -1.0000 | 4.5093 |
HCC1500 | USP7-IN-1 | 72 | 51.9923039456 | 0.4861 | 0.0630 | 130.5080 | -1.0000 | 1.1937 |
MDA-MB-361 | HBX19818 | 72 | 20.1726714877 | -0.3872 | 0.0630 | 34.0507 | -1.0000 | 2.0985 |
BT-20 | HBX19818 | 72 | 30.8921915642 | -0.2433 | 0.0631 | 35.1813 | -0.4578 | 5.0000 |
HCC1428 | STK547622 | 72 | inf | 0.8677 | 0.0634 | 0.0000 | 0.9587 | 0.0100 |
BT-20 | ML-323 | 72 | 211.396631725 | 0.7311 | 0.0653 | 1563.4058 | -1.0000 | 0.5491 |
SK-BR-3 | ML-323 | 72 | 71.5457262907 | 0.6083 | 0.0659 | 250.9976 | -1.0000 | 0.8753 |
HCC1428 | USP7-IN-1 | 72 | inf | 0.6846 | 0.0667 | 0.0000 | 0.9252 | 0.0100 |
PDX1258 | USP7-IN-1 | 72 | inf | 0.8007 | 0.0688 | 0.0000 | 0.9245 | 0.0100 |
PDXHCI002 | USP7-IN-1 | 72 | inf | 0.8827 | 0.0691 | 0.0000 | 0.9313 | 0.0100 |
PDX1258 | z-VAE(OMe)-fmk | 72 | inf | 0.9262 | 0.0692 | 0.0000 | 0.9516 | 0.0100 |
HCC202 | Doxycycline | 72 | 41.0834372075 | 0.2347 | 0.0694 | 58.6649 | -1.0000 | 3.0839 |
T47D | 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one | 72 | inf | 0.9421 | 0.0700 | 0.0000 | 0.9383 | 0.0100 |
PDXHCI002 | IU1 | 72 | inf | 0.7347 | 0.0713 | 0.0000 | 0.9096 | 0.0100 |
HCC202 | HY-17542 | 72 | 68.7359336666 | 0.6087 | 0.0718 | 43.2417 | 0.3314 | 2.3458 |
MDA-MB-231 | SB1-F-22 | 72 | inf | 0.7278 | 0.0733 | 6.1857 | 0.7300 | 3.3947 |
HCC1937 | Spautin-1 | 72 | inf | 0.6302 | 0.0761 | 13.9030 | 0.5336 | 0.8715 |
MCF 10A | Spautin-1 | 72 | inf | 0.7020 | 0.0777 | 4.4596 | 0.7090 | 1.5877 |