Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 2 of 2: Calculated dose response metrics. - Dataset (ID:20351)
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Cell | Small Molecule | Treatment Duration | GR50 | GRmax | GR_AOC | GEC50 | GRinf | hGR |
---|---|---|---|---|---|---|---|---|
SK-BR-3 | ML-323 | 72 | 71.5457262907 | 0.6083 | 0.0659 | 250.9976 | -1.0000 | 0.8753 |
BT-549 | ML-323 | 72 | 74.3999913582 | 0.5763 | 0.0892 | 442.2433 | -1.0000 | 0.6164 |
BT-549 | HY-17541A | 72 | 16.8403527969 | -0.5863 | 0.1928 | 28.1688 | -1.0000 | 2.1356 |
HCC202 | HBX19818 | 72 | 15.8528818617 | -0.3562 | 0.1986 | 34.9884 | -1.0000 | 1.3877 |
BT-549 | HBX19818 | 72 | 28.4956034945 | -0.3396 | 0.1206 | 40.2238 | -1.0000 | 3.1871 |
SK-BR-3 | Doxycycline | 72 | 30.0303971358 | 0.1295 | 0.1243 | 58.5093 | -1.0000 | 1.6472 |
SK-BR-3 | Pimozide | 72 | 4.05486946769 | -0.5520 | 0.4336 | 12.8412 | -1.0000 | 0.9530 |
BT-549 | USP7-IN-1 | 72 | 94.531181628 | 0.8209 | 0.0177 | 166.1357 | -1.0000 | 1.9483 |
T47D | USP7-IN-1 | 72 | 35.2358506575 | 0.3921 | 0.1491 | 300.7608 | -1.0000 | 0.5124 |
T47D | GW7647 | 72 | 29.2962645783 | -0.3773 | 0.0975 | 40.0903 | -1.0000 | 3.5024 |
T47D | HBX19818 | 72 | 19.8447349854 | -0.2828 | 0.1712 | 37.7631 | -1.0000 | 1.7075 |
T47D | HY-17541A | 72 | 6.09725713645 | -0.5568 | 0.3223 | 17.5481 | -1.0000 | 1.0393 |
T47D | HY-17542 | 72 | 60.7583842474 | 0.5918 | 0.0384 | 120.2191 | -1.0000 | 1.6099 |
MCF7 | ML-323 | 72 | 34.9041902184 | 0.3934 | 0.1213 | 138.0045 | -1.0000 | 0.7992 |
HCC202 | Doxycycline | 72 | 41.0834372075 | 0.2347 | 0.0694 | 58.6649 | -1.0000 | 3.0839 |
HCC202 | Mitoxantrone | 72 | 0.00434457297625 | -0.7112 | 1.2184 | 0.1443 | -1.0000 | 0.3136 |
BT-20 | ML-323 | 72 | 211.396631725 | 0.7311 | 0.0653 | 1563.4058 | -1.0000 | 0.5491 |
Hs 578T | ML-323 | 72 | 133.678939825 | 0.6153 | 0.1131 | 2077.0523 | -1.0000 | 0.4005 |
Hs 578T | SB1-F-22 | 72 | 48.629206693 | 0.4746 | 0.0557 | 108.1899 | -1.0000 | 1.3738 |
T47D | Mitoxantrone | 72 | 5.66232793817e-05 | -0.4434 | 1.1468 | 0.0899 | -1.0000 | 0.1491 |
MCF 10A | HBX19818 | 72 | 32.2419133513 | -0.1889 | 0.1089 | 44.8110 | -1.0000 | 3.3374 |
T47D | Pimozide | 72 | 7.11853496187 | -0.5532 | 0.3575 | 16.3429 | -1.0000 | 1.3219 |