Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 1 of 2: Normalized growth rate inhibition values. - Dataset (ID:20350)
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Cell | Small Molecule | Small Mol Concentration (uM) | Mean Normalized Growth Rate Inhibition (GR) Value | Increased Fraction Dead |
---|---|---|---|---|
PDX1258 | STK547622 | 50.0 | 1.0771 | -0.01070 |
PDX1258 | Trifluoperazine | 0.009992797 | 0.9425 | 0.00396 |
PDX1258 | Trifluoperazine | 0.0316 | 0.9126 | 0.03357 |
PDX1258 | Trifluoperazine | 0.099927974 | 0.9621 | 0.01456 |
PDX1258 | Trifluoperazine | 0.316 | 0.8928 | 0.02567 |
PDX1258 | Trifluoperazine | 0.999279741 | 0.9155 | 0.02634 |
PDX1258 | Trifluoperazine | 3.16 | 0.8782 | 0.00782 |
PDX1258 | Trifluoperazine | 9.992797406 | 0.4335 | 0.14169 |
PDX1258 | Trifluoperazine | 31.6 | -0.5938 | 0.55964 |
PDX1258 | Trifluoperazine | 50.0 | -0.6331 | 0.57632 |
PDX1258 | Vialinin A | 0.009992797 | 1.0468 | -0.00628 |
PDX1258 | Vialinin A | 0.0316 | 1.1319 | -0.00961 |
PDX1258 | Vialinin A | 0.099927974 | 1.0008 | -0.00722 |
PDX1258 | Vialinin A | 0.316 | 1.0682 | -0.01120 |
PDX1258 | Vialinin A | 0.999279741 | 1.1541 | -0.02261 |
PDX1258 | Vialinin A | 3.16 | 1.0973 | -0.05502 |
PDX1258 | Vialinin A | 9.992797406 | 0.6609 | 0.03184 |
PDX1258 | Vialinin A | 31.6 | -0.0391 | 0.21872 |
PDX1258 | Vialinin A | 50.0 | -0.2326 | 0.33825 |
PDX1258 | Degrasyn | 0.009992797 | 1.0882 | -0.00116 |
PDX1258 | Degrasyn | 0.0316 | 0.8294 | 0.02042 |
PDX1258 | Degrasyn | 0.099927974 | 1.0404 | -0.00376 |
PDX1258 | Degrasyn | 0.316 | 0.9669 | 0.00808 |
PDX1258 | Degrasyn | 0.999279741 | 0.9419 | 0.08331 |
PDX1258 | Degrasyn | 3.16 | 0.0039 | 0.39581 |