Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 1 of 2: Normalized growth rate inhibition values. - Dataset (ID:20350)
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Cell | Small Molecule | Small Mol Concentration (uM) | Mean Normalized Growth Rate Inhibition (GR) Value | Increased Fraction Dead |
---|---|---|---|---|
T47D | Degrasyn | 0.999279741 | 0.8580 | 0.03874 |
T47D | Degrasyn | 3.16 | -0.1193 | 0.32597 |
T47D | Degrasyn | 9.992797406 | -0.2534 | 0.34895 |
T47D | Degrasyn | 31.6 | -0.5909 | 0.66409 |
T47D | Degrasyn | 50.0 | -0.6099 | 0.54226 |
T47D | Sepantronium | 0.009992797 | 0.8293 | 0.01938 |
T47D | Sepantronium | 0.0316 | 0.3906 | 0.10843 |
T47D | Sepantronium | 0.099927974 | -0.1148 | 0.37177 |
T47D | Sepantronium | 0.316 | -0.3868 | 0.55892 |
T47D | Sepantronium | 0.999279741 | -0.4952 | 0.64682 |
T47D | Sepantronium | 3.16 | -0.5103 | 0.67080 |
T47D | Sepantronium | 9.992797406 | -0.5487 | 0.65344 |
T47D | Sepantronium | 31.6 | -0.5405 | 0.64337 |
T47D | Sepantronium | 50.0 | -0.5680 | 0.47989 |
T47D | z-VAE(OMe)-fmk | 0.009992797 | 1.0454 | -0.00530 |
T47D | z-VAE(OMe)-fmk | 0.0316 | 0.9808 | -0.00714 |
T47D | z-VAE(OMe)-fmk | 0.099927974 | 0.9913 | -0.00648 |
T47D | z-VAE(OMe)-fmk | 0.316 | 0.9437 | -0.00573 |
T47D | z-VAE(OMe)-fmk | 0.999279741 | 1.0055 | -0.00708 |
T47D | z-VAE(OMe)-fmk | 3.16 | 0.9302 | -0.00891 |
T47D | z-VAE(OMe)-fmk | 9.992797406 | 0.9746 | -0.00420 |
T47D | z-VAE(OMe)-fmk | 31.6 | 0.9556 | -0.00497 |
T47D | z-VAE(OMe)-fmk | 50.0 | 0.9468 | -0.00497 |