Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
HCC1428 | Cediranib | 0.0031623 | VEGFR/cKIT | RTK | 1.0052 | -0.00342 |
HCC1428 | Cediranib | 0.01 | VEGFR/cKIT | RTK | 1.0350 | -0.00540 |
HCC1428 | Cediranib | 0.031623 | VEGFR/cKIT | RTK | 0.9364 | -0.00305 |
HCC1428 | Cediranib | 0.1 | VEGFR/cKIT | RTK | 0.9429 | -0.00293 |
HCC1428 | Cediranib | 0.31623 | VEGFR/cKIT | RTK | 0.9279 | 0.00033 |
HCC1428 | Cediranib | 1.0 | VEGFR/cKIT | RTK | 0.7957 | 0.00284 |
HCC1428 | Cediranib | 3.1623 | VEGFR/cKIT | RTK | 0.5526 | 0.04094 |
HCC1428 | Cediranib | 10.0 | VEGFR/cKIT | RTK | -0.5502 | 0.53304 |
HCC1428 | Cabozantinib | 0.001 | VEGFR2/MET | RTK | 1.0383 | -0.00446 |
HCC1428 | Cabozantinib | 0.0031623 | VEGFR2/MET | RTK | 1.0360 | -0.00390 |
HCC1428 | Cabozantinib | 0.01 | VEGFR2/MET | RTK | 1.0784 | -0.00314 |
HCC1428 | Cabozantinib | 0.031623 | VEGFR2/MET | RTK | 1.0983 | -0.00483 |
HCC1428 | Cabozantinib | 0.1 | VEGFR2/MET | RTK | 0.9806 | -0.00580 |
HCC1428 | Cabozantinib | 0.31623 | VEGFR2/MET | RTK | 1.0072 | -0.00615 |
HCC1428 | Cabozantinib | 1.0 | VEGFR2/MET | RTK | 0.9940 | 0.00009 |
HCC1428 | Cabozantinib | 3.1623 | VEGFR2/MET | RTK | 0.8842 | -0.00155 |
HCC1428 | Cabozantinib | 10.0 | VEGFR2/MET | RTK | 0.6310 | 0.02239 |
HME1 | Abemaciclib | 0.001 | CDK4/6 | Cell cycle | 1.0652 | 0.00103 |
HME1 | Abemaciclib | 0.0031623 | CDK4/6 | Cell cycle | 0.9991 | -0.00594 |
HME1 | Abemaciclib | 0.01 | CDK4/6 | Cell cycle | 0.8808 | -0.00310 |
HME1 | Abemaciclib | 0.031623 | CDK4/6 | Cell cycle | 0.7233 | 0.00199 |
HME1 | Abemaciclib | 0.1 | CDK4/6 | Cell cycle | 0.5801 | 0.00750 |
HME1 | Abemaciclib | 0.31623 | CDK4/6 | Cell cycle | 0.4360 | 0.00857 |
HME1 | Abemaciclib | 1.0 | CDK4/6 | Cell cycle | 0.2792 | 0.03205 |
HME1 | Abemaciclib | 3.1623 | CDK4/6 | Cell cycle | 0.1407 | 0.04004 |