Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
HCC1428 | Taselisib | 0.001 | PI3Ka, g, d | PI3K/mTOR | 1.0305 | 0.00006 |
HCC1428 | Taselisib | 0.0031623 | PI3Ka, g, d | PI3K/mTOR | 0.9700 | 0.00244 |
HCC1428 | Taselisib | 0.01 | PI3Ka, g, d | PI3K/mTOR | 1.0865 | 0.00596 |
HCC1428 | Taselisib | 0.031623 | PI3Ka, g, d | PI3K/mTOR | 0.9905 | 0.00082 |
HCC1428 | Taselisib | 0.1 | PI3Ka, g, d | PI3K/mTOR | 0.8814 | 0.01245 |
HCC1428 | Taselisib | 0.31623 | PI3Ka, g, d | PI3K/mTOR | 0.8845 | 0.00355 |
HCC1428 | Taselisib | 1.0 | PI3Ka, g, d | PI3K/mTOR | 0.9055 | 0.01012 |
HCC1428 | Taselisib | 3.1623 | PI3Ka, g, d | PI3K/mTOR | 0.5655 | 0.02918 |
HCC1428 | Taselisib | 10.0 | PI3Ka, g, d | PI3K/mTOR | 0.1734 | 0.10781 |
HCC1428 | TGX221 | 0.001 | PI3Kb | PI3K/mTOR | 1.1327 | 0.00456 |
HCC1428 | TGX221 | 0.0031623 | PI3Kb | PI3K/mTOR | 0.9202 | 0.00052 |
HCC1428 | TGX221 | 0.01 | PI3Kb | PI3K/mTOR | 1.0763 | 0.00096 |
HCC1428 | TGX221 | 0.031623 | PI3Kb | PI3K/mTOR | 1.0395 | 0.00689 |
HCC1428 | TGX221 | 0.1 | PI3Kb | PI3K/mTOR | 1.0296 | 0.00101 |
HCC1428 | TGX221 | 0.31623 | PI3Kb | PI3K/mTOR | 0.9631 | -0.00155 |
HCC1428 | TGX221 | 1.0 | PI3Kb | PI3K/mTOR | 1.0406 | 0.00158 |
HCC1428 | TGX221 | 3.1623 | PI3Kb | PI3K/mTOR | 0.9333 | 0.00032 |
HCC1428 | TGX221 | 10.0 | PI3Kb | PI3K/mTOR | 0.7695 | 0.01533 |
HCC1428 | Torin2 | 0.0001 | mTOR/ATM/ATR | PI3K/mTOR | 0.9850 | 0.00698 |
HCC1428 | Torin2 | 0.00031623 | mTOR/ATM/ATR | PI3K/mTOR | 1.0780 | -0.00215 |
HCC1428 | Torin2 | 0.001 | mTOR/ATM/ATR | PI3K/mTOR | 1.0841 | 0.00186 |
HCC1428 | Torin2 | 0.0031623 | mTOR/ATM/ATR | PI3K/mTOR | 0.8025 | 0.00662 |
HCC1428 | Torin2 | 0.01 | mTOR/ATM/ATR | PI3K/mTOR | 0.5681 | 0.02550 |
HCC1428 | Torin2 | 0.031623 | mTOR/ATM/ATR | PI3K/mTOR | 0.2565 | 0.05576 |
HCC1428 | Torin2 | 0.1 | mTOR/ATM/ATR | PI3K/mTOR | 0.1365 | 0.08363 |