Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
COLO 858 Vemurafenib 0.3160
uM
48
hr
2 1202 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 368.53 NGFR rabbit IgG(H+L) / donkey NGFR 150.06
Colo858-B2-rep2
A4
COLO 858 Vemurafenib 0.3160
uM
48
hr
2 1374 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 335.96 NGFR rabbit IgG(H+L) / donkey NGFR 155.43
Colo858-B2-rep2
A5
COLO 858 Vemurafenib 0.3160
uM
48
hr
2 949 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 432.52 NGFR rabbit IgG(H+L) / donkey NGFR 134.87
Colo858-B2-rep2
A6
COLO 858 Vemurafenib 0.3160
uM
48
hr
2 964 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 357.17 NGFR rabbit IgG(H+L) / donkey NGFR 140.07
Colo858-B2-rep2
A7
COLO 858 Vemurafenib 0.3160
uM
48
hr
2 1020 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 404.61 NGFR rabbit IgG(H+L) / donkey NGFR 144.69
Colo858-B2-rep2
A8
COLO 858 Vemurafenib 0.3160
uM
48
hr
2 1359 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 394.62 NGFR rabbit IgG(H+L) / donkey NGFR 149.61
Colo858-B2-rep2
A9
COLO 858 Vemurafenib Olaparib 0.3160 0.1067
uM
48
hr
2 2065 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 297.06 NGFR rabbit IgG(H+L) / donkey NGFR 150.99
Colo858-B2-rep2
B2
COLO 858 Vemurafenib Iniparib 0.3160 0.1067
uM
48
hr
2 1737 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 342.50 NGFR rabbit IgG(H+L) / donkey NGFR 168.06
Colo858-B2-rep2
B3
COLO 858 Vemurafenib CTB 0.3160 0.1067
uM
48
hr
2 2165 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 297.22 NGFR rabbit IgG(H+L) / donkey NGFR 163.28
Colo858-B2-rep2
B4
COLO 858 Vemurafenib Rocilinostat 0.3160 0.1067
uM
48
hr
2 2119 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 332.77 NGFR rabbit IgG(H+L) / donkey NGFR 180.07
Colo858-B2-rep2
B5
COLO 858 Vemurafenib GSK-J1 0.3160 0.1067
uM
48
hr
2 1949 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 408.18 NGFR rabbit IgG(H+L) / donkey NGFR 166.40
Colo858-B2-rep2
B6
COLO 858 Vemurafenib PFI-1 0.3160 0.1067
uM
48
hr
2 2090 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 400.42 NGFR rabbit IgG(H+L) / donkey NGFR 145.17
Colo858-B2-rep2
B7
COLO 858 Vemurafenib UNC669 0.3160 0.1067
uM
48
hr
2 1966 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 419.20 NGFR rabbit IgG(H+L) / donkey NGFR 177.46
Colo858-B2-rep2
B8
COLO 858 Vemurafenib Veliparib 0.3160 0.1067
uM
48
hr
2 2385 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 352.61 NGFR rabbit IgG(H+L) / donkey NGFR 183.60
Colo858-B2-rep2
C2
COLO 858 Vemurafenib Rucaparib 0.3160 0.1067
uM
48
hr
2 2779 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 314.05 NGFR rabbit IgG(H+L) / donkey NGFR 173.73
Colo858-B2-rep2
C3
COLO 858 Vemurafenib Belinostat 0.3160 0.1067
uM
48
hr
2 796 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 190.45 NGFR rabbit IgG(H+L) / donkey NGFR 129.48
Colo858-B2-rep2
C4
COLO 858 Vemurafenib Selisistat 0.3160 0.1067
uM
48
hr
2 2910 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 357.93 NGFR rabbit IgG(H+L) / donkey NGFR 146.71
Colo858-B2-rep2
C5
COLO 858 Vemurafenib GSK-J2 0.3160 0.1067
uM
48
hr
2 2915 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 358.92 NGFR rabbit IgG(H+L) / donkey NGFR 159.25
Colo858-B2-rep2
C6
COLO 858 Vemurafenib (+)-JQ1 0.3160 0.1067
uM
48
hr
2 2000 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 144.50 NGFR rabbit IgG(H+L) / donkey NGFR 27.98
Colo858-B2-rep2
C7
COLO 858 Vemurafenib UNC1215 0.3160 0.1067
uM
48
hr
2 2912 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 347.33 NGFR rabbit IgG(H+L) / donkey NGFR 170.30
Colo858-B2-rep2
C8
COLO 858 Vemurafenib Vorinostat 0.3160 0.1067
uM
48
hr
2 1954 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 264.42 NGFR rabbit IgG(H+L) / donkey NGFR 180.44
Colo858-B2-rep2
D2
COLO 858 Vemurafenib JW55 0.3160 0.1067
uM
48
hr
2 2613 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 358.73 NGFR rabbit IgG(H+L) / donkey NGFR 151.57
Colo858-B2-rep2
D3
COLO 858 Vemurafenib Entinostat 0.3160 0.1067
uM
48
hr
2 3440 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 282.63 NGFR rabbit IgG(H+L) / donkey NGFR 158.24
Colo858-B2-rep2
D4
COLO 858 Vemurafenib AGK2 0.3160 0.1067
uM
48
hr
2 2858 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 305.97 NGFR rabbit IgG(H+L) / donkey NGFR 137.70
Colo858-B2-rep2
D5
COLO 858 Vemurafenib GSK-J4 0.3160 0.1067
uM
48
hr
2 3387 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 368.22 NGFR rabbit IgG(H+L) / donkey NGFR 158.47
Colo858-B2-rep2
D6