5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | MWCL.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 19.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 16.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -2.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -1.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | 2.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | -31.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | 7.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | 12.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | 2.4 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | -25.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | -2.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 5.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | eEF2K | YIKYNSNSGFVR | ATP | -21.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | eEF2K | YIKYNSNSGFVR | ATP | -19.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | 23.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | 1 | uM | |
| 5z-7-oxozeaenol | BCWM.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | 27.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | -9.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP Loop | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP Loop | 2.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ILK | WQGNDIVVKVLK | Lys1 | -10.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ILK | WQGNDIVVKVLK | Lys1 | 3.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 3.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | -3.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | RIPK2 | VQVAVKHLHIHTPLLDSER | Lys1 | 11.1 | 1 | uM |