WZ3105 KiNativ -- single dose experiment - Dataset (ID:20253)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| WZ3105 | THP-1 | MK14 | QELNKTIWEVPER | Protein Kinase Domain | 18.5 | 1 | uM |
| WZ3105 | THP-1 | CDK9 | DMKAANVLITR | Lys2 | 23.4 | 1 | uM |
| WZ3105 | THP-1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -1.9 | 1 | uM |
| WZ3105 | THP-1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 6.5 | 1 | uM |
| WZ3105 | THP-1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 12.2 | 1 | uM |
| WZ3105 | THP-1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 44.9 | 1 | uM |
| WZ3105 | THP-1 | CDK13 | DIKCSNILLNNR | Lys2 | 26.6 | 1 | uM |
| WZ3105 | THP-1 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 44.3 | 1 | uM |
| WZ3105 | THP-1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | -5.7 | 1 | uM |
| WZ3105 | THP-1 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLKPENLLLASK | Lys2 | 27.6 | 1 | uM |
| WZ3105 | THP-1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | -3.8 | 1 | uM |
| WZ3105 | THP-1 | IKKE,TBK1 | DIKPGNIMR | Lys2 | 0.6 | 1 | uM |
| WZ3105 | THP-1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | -1.5 | 1 | uM |
| WZ3105 | THP-1 | CDK20 | DLKPANLLISASGQLK | Lys2 | 4.9 | 1 | uM |
| WZ3105 | THP-1 | CRK7 | DIKCSNILLNNSGQIK | Lys2 | 35.1 | 1 | uM |
| WZ3105 | THP-1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | -16.9 | 1 | uM |
| WZ3105 | THP-1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | -0.8 | 1 | uM |
| WZ3105 | THP-1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 14.4 | 1 | uM |
| WZ3105 | THP-1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -3.4 | 1 | uM |
| WZ3105 | THP-1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | -10.4 | 1 | uM |
| WZ3105 | THP-1 | CDK5 | DLKPQNLLINR | Lys2 | 39.1 | 1 | uM |
| WZ3105 | THP-1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -2.1 | 1 | uM |
| WZ3105 | THP-1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 64.4 | 1 | uM |
| WZ3105 | THP-1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | 19.0 | 1 | uM |
| WZ3105 | THP-1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 76.4 | 1 | uM |