WZ3105 KiNativ -- single dose experiment - Dataset (ID:20253)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| WZ3105 | THP-1 | CaMK1a | LVAIKCIAK | Lys1 | 0.1 | 1 | uM |
| WZ3105 | THP-1 | eEF2K | YIKYNSNSGFVR | ATP | -0.3 | 1 | uM |
| WZ3105 | THP-1 | IKKE,TBK1 | DIKPGNIMR | Lys2 | 0.6 | 1 | uM |
| WZ3105 | THP-1 | CDK2 | NKLTGEVVALKK | Lys1 | 0.6 | 1 | uM |
| WZ3105 | THP-1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | -0.8 | 1 | uM |
| WZ3105 | THP-1 | MAP2K5 | DVKPSNMLVNTR | Lys2 | -10.0 | 1 | uM |
| WZ3105 | THP-1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -10.2 | 1 | uM |
| WZ3105 | THP-1 | PIK3CD | VNWLAHNVSKDNRQ | ATP | -10.2 | 1 | uM |
| WZ3105 | THP-1 | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | -10.3 | 1 | uM |
| WZ3105 | THP-1 | FER | TSVAVKTCKEDLPQELK | Lys1 | 10.3 | 1 | uM |
| WZ3105 | THP-1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | -10.4 | 1 | uM |
| WZ3105 | THP-1 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | -10.6 | 1 | uM |
| WZ3105 | THP-1 | NEK7 | AACLLDGVPVALKK | Lys1 | -10.7 | 1 | uM |
| WZ3105 | THP-1 | MASTL | LYAVKVVK | Lys1 | -10.8 | 1 | uM |
| WZ3105 | THP-1 | CDK16 | LTDNLVALKEIR | Lys1 | 11.2 | 1 | uM |
| WZ3105 | THP-1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -11.4 | 1 | uM |
| WZ3105 | THP-1 | PDK1 | EYAIKILEK | Lys1 | 11.8 | 1 | uM |
| WZ3105 | THP-1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | 12.0 | 1 | uM |
| WZ3105 | THP-1 | HPK1 | DKVSGDLVALKMVK | Lys1 | 12.1 | 1 | uM |
| WZ3105 | THP-1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 12.2 | 1 | uM |
| WZ3105 | THP-1 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | -12.3 | 1 | uM |
| WZ3105 | THP-1 | PIK3CB | VFGEDSVGVIFKNGDDLR | ATP | -12.9 | 1 | uM |
| WZ3105 | THP-1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -12.9 | 1 | uM |
| WZ3105 | THP-1 | p38a | DLKPSNLAVNEDCELK | Lys2 | 12.9 | 1 | uM |
| WZ3105 | THP-1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | -1.3 | 1 | uM |