WZ3105 KiNativ -- single dose experiment - Dataset (ID:20253)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
WZ3105 THP-1 AMPKa1,AMPKa2
VAVKILNR
Lys1
4.8
1
uM
WZ3105 THP-1 AMPKa1,AMPKa2
DLKPENVLLDAHMNAK
Lys2
-3.8
1
uM
WZ3105 THP-1 ATM
QLVKGRDDLRQDAVMQQVFQMCNTLLQR
ATP
-6.1
1
uM
WZ3105 THP-1 ATR
FYIMMCKPK
ATP
2.4
1
uM
WZ3105 THP-1 AurA
FILALKVLFK
Lys1
4.0
1
uM
WZ3105 THP-1 BRAF
DLKSNNIFLHEDLTVK
Lys2
-1.5
1
uM
WZ3105 THP-1 BTK
YVLDDEYTSSVGSKFPVR
Activation Loop
17.1
1
uM
WZ3105 THP-1 CaMK1a
LVAIKCIAK
Lys1
0.1
1
uM
WZ3105 THP-1 CAMK1D
LFAVKCIPK
Lys1
-2.1
1
uM
WZ3105 THP-1 CaMK2a,CaMK2b,CaMK2d,CaMK2g
DLKPENLLLASK
Lys2
27.6
1
uM
WZ3105 THP-1 KCC2D
IPTGQEYAAKIINTK
Lys1
32.5
1
uM
WZ3105 THP-1 CaMK2g
TSTQEYAAKIINTK
Lys1
46.3
1
uM
WZ3105 THP-1 CaMKK2
LAYNENDNTYYAMKVLSK
Lys1
65.2
1
uM
WZ3105 THP-1 CDK20
DLKPANLLISASGQLK
Lys2
4.9
1
uM
WZ3105 THP-1 CDC2
DLKPQNLLIDDKGTIK
Lys2
-1.9
1
uM
WZ3105 THP-1 CDK11,CDK8
DLKPANILVMGEGPER
Lys2
-16.9
1
uM
WZ3105 THP-1 CDK2
NKLTGEVVALKK
Lys1
0.6
1
uM
WZ3105 THP-1 CDK2
DLKPQNLLINTEGAIK
Lys2
14.4
1
uM
WZ3105 THP-1 CDK4
DLKPENILVTSGGTVK
Lys2
-3.4
1
uM
WZ3105 THP-1 CDK5
NRETHEIVALKR
Lys1
35.7
1
uM
WZ3105 THP-1 CDK5
DLKPQNLLINR
Lys2
39.1
1
uM
WZ3105 THP-1 CDK6
DLKPQNILVTSSGQIK
Lys2
-2.1
1
uM
WZ3105 THP-1 CDK7
DLKPNNLLLDENGVLK
Lys2
64.4
1
uM
WZ3105 THP-1 CDK9
DMKAANVLITR
Lys2
23.4
1
uM
WZ3105 THP-1 ACK
TVSVAVKCLKPDVLSQPEAMDDFIR
Lys1
53.1
1
uM
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