WZ3105 KiNativ -- single dose experiment - Dataset (ID:20253)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| WZ3105 | THP-1 | NEK7 | AACLLDGVPVALKK | Lys1 | -10.7 | 1 | uM |
| WZ3105 | THP-1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 12.2 | 1 | uM |
| WZ3105 | THP-1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | -2.5 | 1 | uM |
| WZ3105 | THP-1 | LATS1 | ALYATKTLR | Lys1 | -90.6 | 1 | uM |
| WZ3105 | THP-1 | RSK1 (Domain 2) | ATNMEYAVKVIDK | Lys1 | 5.2 | 1 | uM |
| WZ3105 | THP-1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | -4.7 | 1 | uM |
| WZ3105 | THP-1 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIKTCK | Lys1 | 74.6 | 1 | uM |
| WZ3105 | THP-1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | 25.2 | 1 | uM |
| WZ3105 | THP-1 | MST1,MST2 | DIKAGNILLNTEGHAK | Lys2 | -3.3 | 1 | uM |
| WZ3105 | THP-1 | CDK13 | DIKCSNILLNNR | Lys2 | 26.6 | 1 | uM |
| WZ3105 | THP-1 | CRK7 | DIKCSNILLNNSGQIK | Lys2 | 35.1 | 1 | uM |
| WZ3105 | THP-1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | 12.0 | 1 | uM |
| WZ3105 | THP-1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 18.3 | 1 | uM |
| WZ3105 | THP-1 | NEK6,NEK7 | DIKPANVFITATGVVK | Lys2 | -9.0 | 1 | uM |
| WZ3105 | THP-1 | IKKE,TBK1 | DIKPGNIMR | Lys2 | 0.6 | 1 | uM |
| WZ3105 | THP-1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 76.4 | 1 | uM |
| WZ3105 | THP-1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | 19.0 | 1 | uM |
| WZ3105 | THP-1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 6.5 | 1 | uM |
| WZ3105 | THP-1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 44.9 | 1 | uM |
| WZ3105 | THP-1 | NEK1 | DIKSQNIFLTK | Lys2 | -6.9 | 1 | uM |
| WZ3105 | THP-1 | NEK9 | DIKTLNIFLTK | Lys2 | 13.2 | 1 | uM |
| WZ3105 | THP-1 | HPK1 | DKVSGDLVALKMVK | Lys1 | 12.1 | 1 | uM |
| WZ3105 | THP-1 | SLK | DLKAGNILFTLDGDIK | Lys2 | 18.7 | 1 | uM |
| WZ3105 | THP-1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -10.2 | 1 | uM |
| WZ3105 | THP-1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | -16.9 | 1 | uM |