WZ3105 KiNativ -- single dose experiment - Dataset (ID:20253)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| WZ3105 | THP-1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | 55.8 | 1 | uM |
| WZ3105 | THP-1 | MER,TYRO3 | KIYSGDYYR | Activation Loop | 23.0 | 1 | uM |
| WZ3105 | THP-1 | NEK3 | SKNIFLTQNGK | Activation Loop | -7.9 | 1 | uM |
| WZ3105 | THP-1 | Wnk1,Wnk2,Wnk4 | IGDLGLATLKR | Activation Loop | -9.3 | 1 | uM |
| WZ3105 | THP-1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | -7.7 | 1 | uM |
| WZ3105 | THP-1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 17.1 | 1 | uM |
| WZ3105 | THP-1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | -7.9 | 1 | uM |
| WZ3105 | THP-1 | PIK3CG | KKPLWLEFK | ATP | 4.4 | 1 | uM |
| WZ3105 | THP-1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | -2.5 | 1 | uM |
| WZ3105 | THP-1 | PIK3CB | VFGEDSVGVIFKNGDDLR | ATP | -12.9 | 1 | uM |
| WZ3105 | THP-1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | -2.9 | 1 | uM |
| WZ3105 | THP-1 | PIK3CD | VNWLAHNVSKDNRQ | ATP | -10.2 | 1 | uM |
| WZ3105 | THP-1 | FYV1 | GGKSGAAFYATEDDRFILK | ATP | -7.7 | 1 | uM |
| WZ3105 | THP-1 | eEF2K | YIKYNSNSGFVR | ATP | -0.3 | 1 | uM |
| WZ3105 | THP-1 | ATM | QLVKGRDDLRQDAVMQQVFQMCNTLLQR | ATP | -6.1 | 1 | uM |
| WZ3105 | THP-1 | DNAPK | EHPFLVKGGEDLR | ATP | -2.9 | 1 | uM |
| WZ3105 | THP-1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | -8.3 | 1 | uM |
| WZ3105 | THP-1 | ATR | FYIMMCKPK | ATP | 2.4 | 1 | uM |
| WZ3105 | THP-1 | PRPK | FLSGLELVKQGAEAR | ATP Loop | 7.1 | 1 | uM |
| WZ3105 | THP-1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 53.1 | 1 | uM |
| WZ3105 | THP-1 | CaMKK2 | LAYNENDNTYYAMKVLSK | Lys1 | 65.2 | 1 | uM |
| WZ3105 | THP-1 | GCK | DTVTSELAAVKIVK | Lys1 | 3.2 | 1 | uM |
| WZ3105 | THP-1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 46.3 | 1 | uM |
| WZ3105 | THP-1 | AurA | FILALKVLFK | Lys1 | 4.0 | 1 | uM |
| WZ3105 | THP-1 | KCC2D | IPTGQEYAAKIINTK | Lys1 | 32.5 | 1 | uM |