Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| Ibrutinib | MWCL.1 | NEK4 | DLKTQNVFLTR | Lys2 | 4.700817535 | 1 | uM |
| Ibrutinib | MWCL.1 | NEK6,NEK7 | DIKPANVFITATGVVK | Lys2 | 5.522288083 | 1 | uM |
| Ibrutinib | MWCL.1 | NEK7 | AACLLDGVPVALKK | Lys1 | -32.79198654 | 1 | uM |
| Ibrutinib | MWCL.1 | NEK8 | DLKTQNILLDK | Lys2 | -10.81498066 | 1 | uM |
| Ibrutinib | MWCL.1 | NEK9 | DIKTLNIFLTK | Lys2 | -0.237961412 | 1 | uM |
| Ibrutinib | MWCL.1 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | -5.216130694 | 1 | uM |
| Ibrutinib | MWCL.1 | p38a | DLKPSNLAVNEDCELK | Lys2 | -7.815671346 | 1 | uM |
| Ibrutinib | MWCL.1 | MK14 | QELNKTIWEVPER | Other | -16.68433891 | 1 | uM |
| Ibrutinib | MWCL.1 | MK11 | QELNKTVWEVPQR | Other | -20.37567449 | 1 | uM |
| Ibrutinib | MWCL.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -15.19530384 | 1 | uM |
| Ibrutinib | MWCL.1 | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | -55.84185365 | 1 | uM |
| Ibrutinib | MWCL.1 | KS6B2 | DLKPENIMLSSQGHIK | Lys2 | -40.33803613 | 1 | uM |
| Ibrutinib | MWCL.1 | PAN3 | VMDPTKILITGK | ATP | -27.71690181 | 1 | uM |
| Ibrutinib | MWCL.1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | 7.894332648 | 1 | uM |
| Ibrutinib | MWCL.1 | PDK1 | EYAIKILEK | Lys1 | 21.2586975 | 1 | uM |
| Ibrutinib | MWCL.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | -31.61111339 | 1 | uM |
| Ibrutinib | MWCL.1 | CDK14 | LVALKVIR | Lys1 | 5.479239804 | 1 | uM |
| Ibrutinib | MWCL.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | ND | 1 | uM |
| Ibrutinib | MWCL.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | -28.9504086 | 1 | uM |
| Ibrutinib | MWCL.1 | PI4KB | VPHTQAVVLNSKDK | ATP | 16.74278657 | 1 | uM |
| Ibrutinib | MWCL.1 | PIK3C2B | VIFKCGDDLRQDMLTLQMIR | ATP | -26.05525385 | 1 | uM |
| Ibrutinib | MWCL.1 | PIK3C3 | TEDGGKYPVIFKHGDDLR | ATP | -3.016899825 | 1 | uM |
| Ibrutinib | MWCL.1 | PIK3CB | VFGEDSVGVIFKNGDDLRQDMLTLQMLR | ATP | -9.461019081 | 1 | uM |
| Ibrutinib | MWCL.1 | PIK3CD | VNWLAHNVSKDNRQ | ATP | 3.806200864 | 1 | uM |
| Ibrutinib | MWCL.1 | PIK3CG | KKPLWLEFK | ATP | -14.51848196 | 1 | uM |