Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
Ibrutinib MWCL.1 NEK7
AACLLDGVPVALKK
Lys1
-32.79198654
1
uM
Ibrutinib BCWM.1 NEK7
AACLLDGVPVALKK
Lys1
11.72564622
1
uM
Ibrutinib BCWM.1 IRAK1
AIQFLHQDSPSLIHGDIKSSNVLLDER
Lys2
-25.21103032
1
uM
Ibrutinib MWCL.1 IRAK1
AIQFLHQDSPSLIHGDIKSSNVLLDER
Lys2
15.56395006
1
uM
Ibrutinib MWCL.1 PIP4K2A
AKELPTLKDNDFINEGQK
ATP
-7.441070191
1
uM
Ibrutinib BCWM.1 PIP4K2A
AKELPTLKDNDFINEGQK
ATP
-5.492209336
1
uM
Ibrutinib BCWM.1 LATS1
ALYATKTLR
Lys1
2.515282486
1
uM
Ibrutinib MWCL.1 LATS1
ALYATKTLR
Lys1
30.59661536
1
uM
Ibrutinib MWCL.1 MLKL
APVAIKVFK
Lys1
2.471839009
1
uM
Ibrutinib BCWM.1 MLKL
APVAIKVFK
Lys1
6.564211837
1
uM
Ibrutinib MWCL.1 PHKg2
ATGHEFAVKIMEVTAER
Lys1
ND
1
uM
Ibrutinib BCWM.1 PHKg2
ATGHEFAVKIMEVTAER
Lys1
-23.59607344
1
uM
Ibrutinib MWCL.1 PLK1
CFEISDADTKEVFAGKIVPK
Lys1
17.91776398
1
uM
Ibrutinib BCWM.1 PLK1
CFEISDADTKEVFAGKIVPK
Lys1
-3.592091178
1
uM
Ibrutinib BCWM.1 PRP4
CNILHADIKPDNILVNESK
Lys2
-8.100671563
1
uM
Ibrutinib MWCL.1 PRP4
CNILHADIKPDNILVNESK
Lys2
-47.19430914
1
uM
Ibrutinib BCWM.1 MST3
DIKAANVLLSEHGEVK
Lys2
-9.956864462
1
uM
Ibrutinib MWCL.1 MST3
DIKAANVLLSEHGEVK
Lys2
4.986768398
1
uM
Ibrutinib BCWM.1 MST4,YSK1
DIKAANVLLSEQGDVK
Lys2
-6.360178382
1
uM
Ibrutinib MWCL.1 MST4,YSK1
DIKAANVLLSEQGDVK
Lys2
-3.600863518
1
uM
Ibrutinib BCWM.1 TAO1,TAOK3
DIKAGNILLTEPGQVK
Lys2
8.693117708
1
uM
Ibrutinib MWCL.1 TAO1,TAOK3
DIKAGNILLTEPGQVK
Lys2
-6.125215797
1
uM
Ibrutinib MWCL.1 MAP3K4
DIKGANIFLTSSGLIK
Lys2
-8.019926684
1
uM
Ibrutinib BCWM.1 MAP3K4
DIKGANIFLTSSGLIK
Lys2
-6.705973934
1
uM
Ibrutinib BCWM.1 HPK1
DIKGANILINDAGEVR
Lys2
8.152400611
1
uM
  • Page 1 of 16
  • 1 to 25 of 378 records