Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
Ibrutinib | MWCL.1 | NEK7 | AACLLDGVPVALKK | Lys1 | -32.79198654 | 1 | uM |
Ibrutinib | BCWM.1 | NEK7 | AACLLDGVPVALKK | Lys1 | 11.72564622 | 1 | uM |
Ibrutinib | BCWM.1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | -25.21103032 | 1 | uM |
Ibrutinib | MWCL.1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 15.56395006 | 1 | uM |
Ibrutinib | MWCL.1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | -7.441070191 | 1 | uM |
Ibrutinib | BCWM.1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | -5.492209336 | 1 | uM |
Ibrutinib | BCWM.1 | LATS1 | ALYATKTLR | Lys1 | 2.515282486 | 1 | uM |
Ibrutinib | MWCL.1 | LATS1 | ALYATKTLR | Lys1 | 30.59661536 | 1 | uM |
Ibrutinib | MWCL.1 | MLKL | APVAIKVFK | Lys1 | 2.471839009 | 1 | uM |
Ibrutinib | BCWM.1 | MLKL | APVAIKVFK | Lys1 | 6.564211837 | 1 | uM |
Ibrutinib | MWCL.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | ND | 1 | uM |
Ibrutinib | BCWM.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | -23.59607344 | 1 | uM |
Ibrutinib | MWCL.1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | 17.91776398 | 1 | uM |
Ibrutinib | BCWM.1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | -3.592091178 | 1 | uM |
Ibrutinib | BCWM.1 | PRP4 | CNILHADIKPDNILVNESK | Lys2 | -8.100671563 | 1 | uM |
Ibrutinib | MWCL.1 | PRP4 | CNILHADIKPDNILVNESK | Lys2 | -47.19430914 | 1 | uM |
Ibrutinib | BCWM.1 | MST3 | DIKAANVLLSEHGEVK | Lys2 | -9.956864462 | 1 | uM |
Ibrutinib | MWCL.1 | MST3 | DIKAANVLLSEHGEVK | Lys2 | 4.986768398 | 1 | uM |
Ibrutinib | BCWM.1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | -6.360178382 | 1 | uM |
Ibrutinib | MWCL.1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | -3.600863518 | 1 | uM |
Ibrutinib | BCWM.1 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | 8.693117708 | 1 | uM |
Ibrutinib | MWCL.1 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | -6.125215797 | 1 | uM |
Ibrutinib | MWCL.1 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | -8.019926684 | 1 | uM |
Ibrutinib | BCWM.1 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | -6.705973934 | 1 | uM |
Ibrutinib | BCWM.1 | HPK1 | DIKGANILINDAGEVR | Lys2 | 8.152400611 | 1 | uM |