JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JNK-IN-8 | A-375 | TLK2 | YVAVkIHQLNK | Lys1 | 2.0 | 1 | uM |
| JNK-IN-8 | A-375 | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | 9.7 | 1 | uM |
| JNK-IN-8 | A-375 | ABL,ARG | YSLTVAVkTLKEDTMEVEEFLK | Lys1 | -2.7 | 1 | uM |
| JNK-IN-8 | A-375 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | 2.6 | 1 | uM |
| JNK-IN-8 | A-375 | eEF2K | YIkYNSNSGFVRDDNIR | Protein Kinase Domain | 10.0 | 1 | uM |
| JNK-IN-8 | A-375 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -5.4 | 1 | uM |
| JNK-IN-8 | A-375 | WEE1 | YIHSMSLVHMDIkPSNIFISR | Lys2 | -68.7 | 1 | uM |
| JNK-IN-8 | A-375 | MK03 | YIHSANVLHRDLkPSNLLINTTCDLK | Lys2 | 28.3 | 1 | uM |
| JNK-IN-8 | A-375 | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | -18.7 | 1 | uM |
| JNK-IN-8 | A-375 | ILK | WQGNDIVVkVLK | Lys1 | -13.1 | 1 | uM |
| JNK-IN-8 | A-375 | MLTK | WISQDKEVAVKk | Lys1 | -7.8 | 1 | uM |
| JNK-IN-8 | A-375 | M3K2 | VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | 4.6 | 1 | uM |
| JNK-IN-8 | A-375 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 4.3 | 1 | uM |
| JNK-IN-8 | A-375 | CSK | VSDFGLTkEASSTQDTGK | Activation Loop | 23.4 | 1 | uM |
| JNK-IN-8 | A-375 | GCN2_domain2 | VQNKLDGCCYAVkR | Lys1 | 9.0 | 1 | uM |
| JNK-IN-8 | A-375 | PIK4CB | VPHTQAVVLNSkDKAPYLIYVEVLECENFDTTSVPARIPENR | ATP | 10.1 | 1 | uM |
| JNK-IN-8 | A-375 | PI4KB | VPHTQAVVLNSKDkAPYLIYVEVLECENFDTTSVPAR | ATP | 25.0 | 1 | uM |
| JNK-IN-8 | A-375 | PI4KB | VPHTQAVVLNSkDK | ATP | 8.0 | 1 | uM |
| JNK-IN-8 | A-375 | NEK6,NEK7 | VMHRDIkPANVFITATGVVK | Lys2 | 15.5 | 1 | uM |
| JNK-IN-8 | A-375 | PAN3 | VMDPTkILITGK | Protein Kinase Domain | -34.7 | 1 | uM |
| JNK-IN-8 | A-375 | CDC2 | VLHRDLkPQNLLIDDKGTIK | Lys2 | 2.2 | 1 | uM |
| JNK-IN-8 | A-375 | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | -1.7 | 1 | uM |
| JNK-IN-8 | A-375 | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | -30.3 | 1 | uM |
| JNK-IN-8 | A-375 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 1.4 | 1 | uM |
| JNK-IN-8 | A-375 | PI42C | VKELPTLkDMDFLNK | ATP | 1.9 | 1 | uM |