JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
JNK-IN-8 | A-375 | EGFR | IPVAIkELR | Lys1 | 0.1 | 1 | uM |
JNK-IN-8 | A-375 | PRPK | FLSGLELVkQGAEAR | ATP Loop | 0.2 | 1 | uM |
JNK-IN-8 | A-375 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 0.2 | 1 | uM |
JNK-IN-8 | A-375 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | 0.3 | 1 | uM |
JNK-IN-8 | A-375 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 0.4 | 1 | uM |
JNK-IN-8 | A-375 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 0.5 | 1 | uM |
JNK-IN-8 | A-375 | M3K2 | ELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -0.6 | 1 | uM |
JNK-IN-8 | A-375 | KS6B1 | LTDFGLCkESIHDGTVTHTFCGTIEYMAPEILMR | Activation Loop | -0.6 | 1 | uM |
JNK-IN-8 | A-375 | MAP2K1,MAP2K2 | kLIHLEIKPAIR | Lys1 | -0.7 | 1 | uM |
JNK-IN-8 | A-375 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | -0.8 | 1 | uM |
JNK-IN-8 | A-375 | IRAK1 | AIQFLHQDSPSLIHGDIkSSNVLLDER | Lys2 | 0.8 | 1 | uM |
JNK-IN-8 | A-375 | MST3 | DIkAANVLLSEHGEVK | Lys2 | -0.9 | 1 | uM |
JNK-IN-8 | A-375 | KHS1 | NVHTGELAAVkIIK | Lys1 | -0.9 | 1 | uM |
JNK-IN-8 | A-375 | ROCK1 | kLQLELNQER | Other | 10.0 | 1 | uM |
JNK-IN-8 | A-375 | eEF2K | YIkYNSNSGFVRDDNIR | Protein Kinase Domain | 10.0 | 1 | uM |
JNK-IN-8 | A-375 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 10.0 | 1 | uM |
JNK-IN-8 | A-375 | PIK4CB | VPHTQAVVLNSkDKAPYLIYVEVLECENFDTTSVPARIPENR | ATP | 10.1 | 1 | uM |
JNK-IN-8 | A-375 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -10.2 | 1 | uM |
JNK-IN-8 | A-375 | GCK | DIkGANLLLTLQGDVK | Lys2 | 10.4 | 1 | uM |
JNK-IN-8 | A-375 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 10.5 | 1 | uM |
JNK-IN-8 | A-375 | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | 10.6 | 1 | uM |
JNK-IN-8 | A-375 | ATM | QLVkGRDDLRQDAVMQQVFQMCNTLLQR | ATP | 10.6 | 1 | uM |
JNK-IN-8 | A-375 | RSK2_domain2 | DLkPSNILYVDESGNPESIR | Lys2 | 10.7 | 1 | uM |
JNK-IN-8 | A-375 | MST1,MST2 | IHRDIkAGNILLNTEGHAK | Lys2 | -10.9 | 1 | uM |
JNK-IN-8 | A-375 | NDR1 | DTGHVYAMkILR | Lys1 | -10.9 | 1 | uM |