JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JNK-IN-8 A-375 EGFR
IPVAIkELR
Lys1
0.1
1
uM
JNK-IN-8 A-375 PRPK
FLSGLELVkQGAEAR
ATP Loop
0.2
1
uM
JNK-IN-8 A-375 MK03
DLkPSNLLINTTCDLK
Lys2
0.2
1
uM
JNK-IN-8 A-375 MAP3K4
DIkGANIFLTSSGLIK
Lys2
0.3
1
uM
JNK-IN-8 A-375 CDK11,CDK8
DLkPANILVMGEGPER
Lys2
0.4
1
uM
JNK-IN-8 A-375 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
0.5
1
uM
JNK-IN-8 A-375 M3K2
ELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
-0.6
1
uM
JNK-IN-8 A-375 KS6B1
LTDFGLCkESIHDGTVTHTFCGTIEYMAPEILMR
Activation Loop
-0.6
1
uM
JNK-IN-8 A-375 MAP2K1,MAP2K2
kLIHLEIKPAIR
Lys1
-0.7
1
uM
JNK-IN-8 A-375 PHKg2
ATGHEFAVkIMEVTAER
Lys1
-0.8
1
uM
JNK-IN-8 A-375 IRAK1
AIQFLHQDSPSLIHGDIkSSNVLLDER
Lys2
0.8
1
uM
JNK-IN-8 A-375 MST3
DIkAANVLLSEHGEVK
Lys2
-0.9
1
uM
JNK-IN-8 A-375 KHS1
NVHTGELAAVkIIK
Lys1
-0.9
1
uM
JNK-IN-8 A-375 ROCK1
kLQLELNQER
Other
10.0
1
uM
JNK-IN-8 A-375 eEF2K
YIkYNSNSGFVRDDNIR
Protein Kinase Domain
10.0
1
uM
JNK-IN-8 A-375 MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
10.0
1
uM
JNK-IN-8 A-375 PIK4CB
VPHTQAVVLNSkDKAPYLIYVEVLECENFDTTSVPARIPENR
ATP
10.1
1
uM
JNK-IN-8 A-375 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
-10.2
1
uM
JNK-IN-8 A-375 GCK
DIkGANLLLTLQGDVK
Lys2
10.4
1
uM
JNK-IN-8 A-375 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
10.5
1
uM
JNK-IN-8 A-375 GSK3A
DIkPQNLLVDPDTAVLK
Lys2
10.6
1
uM
JNK-IN-8 A-375 ATM
QLVkGRDDLRQDAVMQQVFQMCNTLLQR
ATP
10.6
1
uM
JNK-IN-8 A-375 RSK2_domain2
DLkPSNILYVDESGNPESIR
Lys2
10.7
1
uM
JNK-IN-8 A-375 MST1,MST2
IHRDIkAGNILLNTEGHAK
Lys2
-10.9
1
uM
JNK-IN-8 A-375 NDR1
DTGHVYAMkILR
Lys1
-10.9
1
uM
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