NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
-12.4
0.50
uM
NVP-BHG712 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
3.4
0.50
uM
NVP-BHG712 PC-3 PIP4K2A
AKELPTLkDNDFINEGQK
ATP
-0.5
0.50
uM
NVP-BHG712 PC-3 PIP4K2B
DLPTFkDNDFLNEGQK
ATP
2.1
0.50
uM
NVP-BHG712 PC-3 PI42C
VKELPTLkDMDFLNK
ATP
-15.0
0.50
uM
NVP-BHG712 PC-3 PI42C
ELPTLkDMDFLNK
ATP
8.6
0.50
uM
NVP-BHG712 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
-29.8
0.50
uM
NVP-BHG712 PC-3 FYV1
GGkSGAAFYATEDDRFILK
ATP
65.2
0.50
uM
NVP-BHG712 PC-3 PITSLRE
DLkTSNLLLSHAGILK
Lys2
-7.3
0.50
uM
NVP-BHG712 PC-3 PRKACB
DLkPENLLIDHQGYIQ
Lys2
5.6
0.50
uM
NVP-BHG712 PC-3 PKD3
NIVHCDLkPENVLLASAEPFPQVK
Lys2
-12.5
0.50
uM
NVP-BHG712 PC-3 PKN1
VLLSEFRPSGELFAIkALK
Lys1
-6.5
0.50
uM
NVP-BHG712 PC-3 PKN2
DLkLDNLLLDTEGFVK
Lys2
0.8
0.50
uM
NVP-BHG712 PC-3 PKR
DLkPSNIFLVDTK
Lys2
10.0
0.50
uM
NVP-BHG712 PC-3 PLK1
CFEISDADTKEVFAGkIVPK
Lys1
-14.4
0.50
uM
NVP-BHG712 PC-3 PLK1
DLkLGNLFLNEDLEVK
Lys2
26.3
0.50
uM
NVP-BHG712 PC-3 PRP4
CNILHADIkPDNILVNESK
Lys2
4.5
0.50
uM
NVP-BHG712 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
25.8
0.50
uM
NVP-BHG712 PC-3 QIK
TEVAIkIIDK
Lys1
12.4
0.50
uM
NVP-BHG712 PC-3 RAF1
DMkSNNIFLHEGLTVK
Lys2
8.5
0.50
uM
NVP-BHG712 PC-3 RIPK2
VQVAVkHLHIHTPLLDSER
Lys1
16.3
0.50
uM
NVP-BHG712 PC-3 ROCK1
kLQLELNQER
Other
5.2
0.50
uM
NVP-BHG712 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-12.8
0.50
uM
NVP-BHG712 PC-3 RON
IQCAIkSLSR
Lys1
-2.3
0.50
uM
NVP-BHG712 PC-3 RSK1_domain2
DLkPSNILYVDESGNPECLR
Lys2
3.5
0.50
uM