NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
NVP-BHG712 | PC-3 | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | -12.4 | 0.50 | uM |
NVP-BHG712 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | 3.4 | 0.50 | uM |
NVP-BHG712 | PC-3 | PIP4K2A | AKELPTLkDNDFINEGQK | ATP | -0.5 | 0.50 | uM |
NVP-BHG712 | PC-3 | PIP4K2B | DLPTFkDNDFLNEGQK | ATP | 2.1 | 0.50 | uM |
NVP-BHG712 | PC-3 | PI42C | VKELPTLkDMDFLNK | ATP | -15.0 | 0.50 | uM |
NVP-BHG712 | PC-3 | PI42C | ELPTLkDMDFLNK | ATP | 8.6 | 0.50 | uM |
NVP-BHG712 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | -29.8 | 0.50 | uM |
NVP-BHG712 | PC-3 | FYV1 | GGkSGAAFYATEDDRFILK | ATP | 65.2 | 0.50 | uM |
NVP-BHG712 | PC-3 | PITSLRE | DLkTSNLLLSHAGILK | Lys2 | -7.3 | 0.50 | uM |
NVP-BHG712 | PC-3 | PRKACB | DLkPENLLIDHQGYIQ | Lys2 | 5.6 | 0.50 | uM |
NVP-BHG712 | PC-3 | PKD3 | NIVHCDLkPENVLLASAEPFPQVK | Lys2 | -12.5 | 0.50 | uM |
NVP-BHG712 | PC-3 | PKN1 | VLLSEFRPSGELFAIkALK | Lys1 | -6.5 | 0.50 | uM |
NVP-BHG712 | PC-3 | PKN2 | DLkLDNLLLDTEGFVK | Lys2 | 0.8 | 0.50 | uM |
NVP-BHG712 | PC-3 | PKR | DLkPSNIFLVDTK | Lys2 | 10.0 | 0.50 | uM |
NVP-BHG712 | PC-3 | PLK1 | CFEISDADTKEVFAGkIVPK | Lys1 | -14.4 | 0.50 | uM |
NVP-BHG712 | PC-3 | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | 26.3 | 0.50 | uM |
NVP-BHG712 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | 4.5 | 0.50 | uM |
NVP-BHG712 | PC-3 | PRPK | FLSGLELVkQGAEAR | ATP Loop | 25.8 | 0.50 | uM |
NVP-BHG712 | PC-3 | QIK | TEVAIkIIDK | Lys1 | 12.4 | 0.50 | uM |
NVP-BHG712 | PC-3 | RAF1 | DMkSNNIFLHEGLTVK | Lys2 | 8.5 | 0.50 | uM |
NVP-BHG712 | PC-3 | RIPK2 | VQVAVkHLHIHTPLLDSER | Lys1 | 16.3 | 0.50 | uM |
NVP-BHG712 | PC-3 | ROCK1 | kLQLELNQER | Other | 5.2 | 0.50 | uM |
NVP-BHG712 | PC-3 | ROCK1,ROCK2 | DVkPDNMLLDK | Lys2 | -12.8 | 0.50 | uM |
NVP-BHG712 | PC-3 | RON | IQCAIkSLSR | Lys1 | -2.3 | 0.50 | uM |
NVP-BHG712 | PC-3 | RSK1_domain2 | DLkPSNILYVDESGNPECLR | Lys2 | 3.5 | 0.50 | uM |