NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NVP-BHG712 | PC-3 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | -10.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MST3 | DIkAANVLLSEHGEVK | Lys2 | 13.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | 17.4 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NDR1 | DTGHVYAMkILR | Lys1 | 15.9 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | 13.4 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NDR2 | DIkPDNLLLDAK | Lys2 | -2.2 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NEK1 | DIkSQNIFLTK | Lys2 | 2.7 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NEK4 | DLkTQNVFLTR | Lys2 | 12.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 18.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NEK7 | AACLLDGVPVALkK | Lys1 | 19.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NEK8 | DLkTQNILLDK | Lys2 | -1.8 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 18.2 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NEK9 | TEDDSLVVWkEVDLTR | Lys1 | 3.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | 10.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | OSR1 | DVkAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | 9.1 | 5.00 | uM |
| NVP-BHG712 | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | 90.0 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MK14 | QELNkTIWEVPER | Other | 44.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MK11 | QELNkTVWEVPQR | Other | -114.2 | 5.00 | uM |
| NVP-BHG712 | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | 9.9 | 5.00 | uM |
| NVP-BHG712 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 11.4 | 5.00 | uM |
| NVP-BHG712 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | 14.0 | 5.00 | uM |
| NVP-BHG712 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | 18.4 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PCTAIRE2 | DLkPQNLLINEK | Lys2 | 7.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PCTAIRE2,PCTAIRE3 | SKLTENLVALkEIR | Lys1 | 14.0 | 5.00 | uM |
| NVP-BHG712 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 30.5 | 5.00 | uM |