NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
Lys2
-1.4
 0.50
uM
NVP-BHG712 PC-3 RSK1,RSK2,RSK3_domain1
DLkPENILLDEEGHIK
Lys2
3.3
 0.50
uM
NVP-BHG712 PC-3 RSK1,RSK3_domain2
SkRDPSEEIEILLR
Protein Kinase Domain
-9.1
 0.50
uM
NVP-BHG712 PC-3 RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
7.3
 0.50
uM
NVP-BHG712 PC-3 RSK2 domain1
VLGQGSFGkVFLVK
ATP Loop
20.2
 0.50
uM
NVP-BHG712 PC-3 RSK2_domain2
DLkPSNILYVDESGNPESIR
Lys2
15.2
 0.50
uM
NVP-BHG712 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
-15.5
 0.50
uM
NVP-BHG712 PC-3 RSK4 domain1
DLkPENILLDEIGHIK
Lys2
23.9
 0.50
uM
NVP-BHG712 PC-3 RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
-18.7
 0.50
uM
NVP-BHG712 PC-3 SGK3
FYAVkVLQK
Lys1
3.1
 0.50
uM
NVP-BHG712 PC-3 SLK
ETSVLAAAkVIDTK
Lys1
-14.9
 0.50
uM
NVP-BHG712 PC-3 SLK
DLkAGNILFTLDGDIK
Lys2
6.4
 0.50
uM
NVP-BHG712 PC-3 SMG1
DTVTIHSVGGTITILPTKTkPK
ATP
-8.2
 0.50
uM
NVP-BHG712 PC-3 SNRK
DLkPENVVFFEK
Lys2
8.7
 0.50
uM
NVP-BHG712 PC-3 SRPK1
IIHTDIkPENILLSVNEQYIR
Lys2
-5.5
 0.50
uM
NVP-BHG712 PC-3 SRPK1/2
FVAMkVVK
Lys1
1.2
 0.50
uM
NVP-BHG712 PC-3 STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
3.5
 0.50
uM
NVP-BHG712 PC-3 STLK5
SVkASHILISVDGK
Lys2
17.8
 0.50
uM
NVP-BHG712 PC-3 STLK6
HTPTGTLVTIkITNLENCNEER
Lys1
8.8
 0.50
uM
NVP-BHG712 PC-3 STLK6
SIkASHILISGDGLVTLSGLSHLHSLVK
Lys2
-9.0
 0.50
uM
NVP-BHG712 PC-3 MAP3K7,TAK1
DLkPPNLLLVAGGTVLK
Lys2
-4.5
 0.50
uM
NVP-BHG712 PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
14.0
 0.50
uM
NVP-BHG712 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
17.0
 0.50
uM
NVP-BHG712 PC-3 TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
9.6
 0.50
uM
NVP-BHG712 PC-3 TLK1
YAAVkIHQLNK
Lys1
17.2
 0.50
uM