NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 NEK4
DLkTQNVFLTR
Lys2
11.7
 0.50
uM
NVP-BHG712 PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
18.0
 0.50
uM
NVP-BHG712 PC-3 NEK7
AACLLDGVPVALkK
Lys1
17.2
 0.50
uM
NVP-BHG712 PC-3 NEK8
DLkTQNILLDK
Lys2
17.1
 0.50
uM
NVP-BHG712 PC-3 NEK9
LGDYGLAkK
Activation Loop
0.8
 0.50
uM
NVP-BHG712 PC-3 NEK9
TEDDSLVVWkEVDLTR
Lys1
2.4
 0.50
uM
NVP-BHG712 PC-3 NEK9
DIkTLNIFLTK
Lys2
6.8
 0.50
uM
NVP-BHG712 PC-3 OSR1
DVkAGNILLGEDGSVQIADFGVSAFLATGGDITR
Lys2
3.2
 0.50
uM
NVP-BHG712 PC-3 p38a
DLkPSNLAVNEDCELK
Lys2
90.0
 0.50
uM
NVP-BHG712 PC-3 MK14
QELNkTIWEVPER
Other
47.4
 0.50
uM
NVP-BHG712 PC-3 MK11
QELNkTVWEVPQR
Other
-85.7
 0.50
uM
NVP-BHG712 PC-3 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
9.7
 0.50
uM
NVP-BHG712 PC-3 KS6B1
DLkPENIMLNHQGHVK
Lys2
-22.3
 0.50
uM
NVP-BHG712 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
13.0
 0.50
uM
NVP-BHG712 PC-3 CDK16
LTDNLVALkEIR
Lys1
10.6
 0.50
uM
NVP-BHG712 PC-3 PCTAIRE2
DLkPQNLLINEK
Lys2
-1.8
 0.50
uM
NVP-BHG712 PC-3 PCTAIRE2,PCTAIRE3
SKLTENLVALkEIR
Lys1
-11.7
 0.50
uM
NVP-BHG712 PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
17.7
 0.50
uM
NVP-BHG712 PC-3 CDK14
LVALkVIR
Lys1
-4.2
 0.50
uM
NVP-BHG712 PC-3 CDK14
DLkPQNLLISDTGELK
Lys2
15.3
 0.50
uM
NVP-BHG712 PC-3 PHKg1
DLkPENILLDDNMNIK
Lys2
15.7
 0.50
uM
NVP-BHG712 PC-3 PHKg2
ATGHEFAVkIMEVTAER
Lys1
-26.2
 0.50
uM
NVP-BHG712 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
0.4
 0.50
uM
NVP-BHG712 PC-3 PI4KB
VPHTQAVVLNSkDKAPYLIYVEVLECENFDTTSVPAR
ATP
-12.1
 0.50
uM
NVP-BHG712 PC-3 PIK3C3
TEDGGKYPVIFkHGDDLRQDQLILQIISLMDK
ATP
8.0
 0.50
uM