NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NVP-BHG712 | PC-3 | BCKDK | QLLDDHkDVVTLLAEGLR | Other | 8.0 | 0.05 | uM |
| NVP-BHG712 | PC-3 | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 7.2 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CaMK1a | LVAIkCIAK | Lys1 | -11.2 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CAMK1D | LFAVkCIPK | Lys1 | -6.7 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | -2.8 | 0.05 | uM |
| NVP-BHG712 | PC-3 | KCC2D | IPTGQEYAAkIINTK | Lys1 | 6.7 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 6.3 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CaMK2g | KTSTQEYAAkIINTKK | Lys1 | -12.7 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | -8.1 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDC2 | DLkPQNLLIDDKGTIK | Lys2 | -3.6 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | -4.7 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK2 | NKLTGEVVALKk | Lys1 | 1.8 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK2 | LTGEVVALkK | Lys1 | 1.2 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 7.6 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | 7.5 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK5 | NRETHEIVALkR | Lys1 | 3.0 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 2.0 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK7 | DLkPNNLLLDENGVLK | Lys2 | 7.1 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK9 | DMkAANVLITR | Lys2 | 12.4 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CHK1 | LSkGDGLEFK | Other | 16.9 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CHK2 | VAIkIISK | Lys1 | 10.3 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | -4.1 | 0.05 | uM |
| NVP-BHG712 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | -3.0 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -6.9 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CSK | VSDFGLTkEASSTQDTGK | Activation Loop | 13.9 | 0.05 | uM |