NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NVP-BHG712 | PC-3 | STLK6 | HTPTGTLVTIkITNLENCNEER | Lys1 | 19.5 | 5.00 | uM |
| NVP-BHG712 | PC-3 | STLK6 | SIkASHILISGDGLVTLSGLSHLHSLVK | Lys2 | 2.2 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MAP3K7,TAK1 | DLkPPNLLLVAGGTVLK | Lys2 | 10.7 | 5.00 | uM |
| NVP-BHG712 | PC-3 | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | 10.8 | 5.00 | uM |
| NVP-BHG712 | PC-3 | TAOK2 | DVkAGNILLSEPGLVK | Lys2 | 22.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | 3.9 | 5.00 | uM |
| NVP-BHG712 | PC-3 | TLK1 | YAAVkIHQLNK | Lys1 | 32.1 | 5.00 | uM |
| NVP-BHG712 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -14.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | 12.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | ULK1 | DLkPQNILLSNPAGR | Lys2 | -0.4 | 5.00 | uM |
| NVP-BHG712 | PC-3 | ULK3 | EVVAIKCVAk | Lys1 | 2.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | ULK3 | NISHLDLkPQNILLSSLEKPHLK | Lys2 | 10.2 | 5.00 | uM |
| NVP-BHG712 | PC-3 | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | -21.0 | 5.00 | uM |
| NVP-BHG712 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -0.7 | 5.00 | uM |
| NVP-BHG712 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | 3.3 | 5.00 | uM |
| NVP-BHG712 | PC-3 | YANK3 | DVkPDNILLDER | Lys2 | 5.6 | 5.00 | uM |
| NVP-BHG712 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 91.0 | 5.00 | uM |
| NVP-BHG712 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 7.7 | 5.00 | uM |
| NVP-BHG712 | PC-3 | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 39.9 | 0.50 | uM |
| NVP-BHG712 | PC-3 | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 0.3 | 0.50 | uM |
| NVP-BHG712 | PC-3 | AGK | ATVFLNPAACkGK | ATP | 2.2 | 0.50 | uM |
| NVP-BHG712 | PC-3 | AMPKa1 | IGHYILGDTLGVGTFGkVK | ATP Loop | 2.1 | 0.50 | uM |
| NVP-BHG712 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | -10.3 | 0.50 | uM |
| NVP-BHG712 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -40.9 | 0.50 | uM |
| NVP-BHG712 | PC-3 | AMPKa2 | IGHYVLGDTLGVGTFGkVK | ATP Loop | -17.5 | 0.50 | uM |