NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NVP-BHG712 | PC-3 | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -8.5 | 0.50 | uM |
| NVP-BHG712 | PC-3 | ATR | FYIMMCkPK | ATP | -11.6 | 0.50 | uM |
| NVP-BHG712 | PC-3 | ATR | kAGHHQTAYNALLNAGESR | Protein Kinase Domain | 5.9 | 0.50 | uM |
| NVP-BHG712 | PC-3 | AurA | FILALkVLFK | Lys1 | 14.4 | 0.50 | uM |
| NVP-BHG712 | PC-3 | AurA | DIkPENLLLGSAGELK | Lys2 | 11.2 | 0.50 | uM |
| NVP-BHG712 | PC-3 | AurB | SHFIVALkVLFK | Lys1 | 25.7 | 0.50 | uM |
| NVP-BHG712 | PC-3 | BARK1 | DLkPANILLDEHGHVR | Lys2 | -27.7 | 0.50 | uM |
| NVP-BHG712 | PC-3 | BCKDK | QLLDDHkDVVTLLAEGLR | Other | 3.1 | 0.50 | uM |
| NVP-BHG712 | PC-3 | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 35.7 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CaMK1a | LVAIkCIAK | Lys1 | -12.5 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CAMK1D | LFAVkCIPK | Lys1 | 1.4 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 2.4 | 0.50 | uM |
| NVP-BHG712 | PC-3 | KCC2D | IPTGQEYAAkIINTK | Lys1 | 0.1 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 5.2 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CaMK2g | KTSTQEYAAkIINTKK | Lys1 | -17.9 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | -17.6 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CDC2 | DLkPQNLLIDDKGTIK | Lys2 | -0.5 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 15.1 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CDK2 | NKLTGEVVALKk | Lys1 | -5.7 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CDK2 | LTGEVVALkK | Lys1 | 2.2 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 14.0 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | -15.4 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CDK5 | NRETHEIVALkR | Lys1 | -11.7 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 11.0 | 0.50 | uM |
| NVP-BHG712 | PC-3 | CDK7 | DLkPNNLLLDENGVLK | Lys2 | 20.8 | 0.50 | uM |