NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

 Full screen view
Filter results: >>>>
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-8.6
 0.50
uM
NVP-BHG712 PC-3 TLK2
YVAVkIHQLNK
Lys1
-12.7
 0.50
uM
NVP-BHG712 PC-3 ULK1
DLkPQNILLSNPAGR
Lys2
-2.4
 0.50
uM
NVP-BHG712 PC-3 ULK3
EVVAIKCVAk
Lys1
-2.7
 0.50
uM
NVP-BHG712 PC-3 ULK3
NISHLDLkPQNILLSSLEKPHLK
Lys2
-7.1
 0.50
uM
NVP-BHG712 PC-3 Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-1.2
 0.50
uM
NVP-BHG712 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-11.5
 0.50
uM
NVP-BHG712 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
-10.3
 0.50
uM
NVP-BHG712 PC-3 YANK3
DVkPDNILLDER
Lys2
4.2
 0.50
uM
NVP-BHG712 PC-3 MLTK
WISQDKEVAVKk
Lys1
92.5
 0.50
uM
NVP-BHG712 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
15.9
 0.50
uM
NVP-BHG712 PC-3 ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
12.2
 0.05
uM
NVP-BHG712 PC-3 ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
-22.3
 0.05
uM
NVP-BHG712 PC-3 AGK
ATVFLNPAACkGK
ATP
-2.0
 0.05
uM
NVP-BHG712 PC-3 AMPKa1
IGHYILGDTLGVGTFGkVK
ATP Loop
-4.6
 0.05
uM
NVP-BHG712 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
-1.6
 0.05
uM
NVP-BHG712 PC-3 AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
20.6
 0.05
uM
NVP-BHG712 PC-3 AMPKa2
IGHYVLGDTLGVGTFGkVK
ATP Loop
-6.2
 0.05
uM
NVP-BHG712 PC-3 ARAF
DLkSNNIFLHEGLTVK
Lys2
-15.6
 0.05
uM
NVP-BHG712 PC-3 ATR
FYIMMCkPK
ATP
3.3
 0.05
uM
NVP-BHG712 PC-3 ATR
kAGHHQTAYNALLNAGESR
Protein Kinase Domain
5.3
 0.05
uM
NVP-BHG712 PC-3 AurA
FILALkVLFK
Lys1
9.0
 0.05
uM
NVP-BHG712 PC-3 AurA
DIkPENLLLGSAGELK
Lys2
10.2
 0.05
uM
NVP-BHG712 PC-3 AurB
SHFIVALkVLFK
Lys1
21.0
 0.05
uM
NVP-BHG712 PC-3 BARK1
DLkPANILLDEHGHVR
Lys2
-26.5
 0.05
uM