XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | PC-3 | PRPK | FLSGLELVkQGAEAR | ATP Loop | 9.7 | 10 | uM |
| XMD8-92 | HeLa | AurB | SHFIVALkVLFK | Lys1 | 9.7 | 10 | uM |
| XMD8-92 | HeLa | LOK | NKETGALAAAkVIETK | Lys1 | -9.7 | 10 | uM |
| XMD8-92 | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | -9.7 | 10 | uM |
| XMD8-92 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 96.0 | 10 | uM |
| XMD8-92 | PC-3 | GCN2 | LDGCCYAVkR | Lys1 | 9.4 | 10 | uM |
| XMD8-92 | PC-3 | MST1,MST2 | DIkAGNILLNTEGHAK | Lys2 | -9.4 | 10 | uM |
| XMD8-92 | PC-3 | PI42C | ELPTLkDMDFLNK | ATP | 9.3 | 10 | uM |
| XMD8-92 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | 9.3 | 10 | uM |
| XMD8-92 | PC-3 | SLK | ETSVLAAAkVIDTK | Lys1 | -9.3 | 10 | uM |
| XMD8-92 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | -9.3 | 10 | uM |
| XMD8-92 | HeLa | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 9.2 | 10 | uM |
| XMD8-92 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 9.2 | 10 | uM |
| XMD8-92 | HeLa | BTK | GQYDVAIkMIK | Lys1 | -9.2 | 10 | uM |
| XMD8-92 | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | -9.2 | 10 | uM |
| XMD8-92 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | -9.2 | 10 | uM |
| XMD8-92 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 9.1 | 10 | uM |
| XMD8-92 | HeLa | MAST2,MAST4 | DLkPDNLLVTSMGHIK | Lys2 | 9.1 | 10 | uM |
| XMD8-92 | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | 9.0 | 10 | uM |
| XMD8-92 | HeLa | MASTL | LYAVkVVK | Lys1 | 8.9 | 10 | uM |
| XMD8-92 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 8.9 | 10 | uM |
| XMD8-92 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | 8.8 | 10 | uM |
| XMD8-92 | PC-3 | MK11 | QELNkTVWEVPQR | Other | 8.8 | 10 | uM |
| XMD8-92 | HeLa | SGK3 | FYAVkVLQK | Lys1 | -8.8 | 10 | uM |
| XMD8-92 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | -8.6 | 10 | uM |