XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
40.4
10
uM
XMD8-92 PC-3 AGK
ATVFLNPAACkGK
ATP
-18.4
10
uM
XMD8-92 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
-16.3
10
uM
XMD8-92 PC-3 AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
11.7
10
uM
XMD8-92 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
6.7
10
uM
XMD8-92 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
3.9
10
uM
XMD8-92 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
-15.6
10
uM
XMD8-92 HeLa ATR
FYIMMCkPK
ATP
-5.7
10
uM
XMD8-92 PC-3 ATR
FYIMMCkPK
ATP
6.1
10
uM
XMD8-92 HeLa BRAF
DLkSNNIFLHEDLTVK
Lys2
-15.5
10
uM
XMD8-92 HeLa CaMK1a
LVAIkCIAK
Lys1
-6.3
10
uM
XMD8-92 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
2.7
10
uM
XMD8-92 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
7.2
10
uM
XMD8-92 PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
1.6
10
uM
XMD8-92 PC-3 CDK10
DLkVSNLLMTDK
Lys2
-8.1
10
uM
XMD8-92 PC-3 CDK11,CDK8
DLkPANILVMGEGPER
Lys2
2.8
10
uM
XMD8-92 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
-18.6
10
uM
XMD8-92 PC-3 CDK2
DLkPQNLLINTEGAIK
Lys2
9.2
10
uM
XMD8-92 PC-3 CDK5
NRETHEIVALkR
Lys1
1.0
10
uM
XMD8-92 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
-11.2
10
uM
XMD8-92 PC-3 CDK9
DMkAANVLITR
Lys2
-16.1
10
uM
XMD8-92 PC-3 CHK2
VAIkIISK
Lys1
2.6
10
uM
XMD8-92 PC-3 KC1A
DIkPDNFLMGIGR
Lys2
-1.7
10
uM
XMD8-92 PC-3 CK1d,CK1e
DVkPDNFLMGLGKK
Lys2
-5.8
10
uM
XMD8-92 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
-28.7
10
uM
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