XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | -26.2 | 10 | uM |
| XMD8-92 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 6.7 | 10 | uM |
| XMD8-92 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | -7.2 | 10 | uM |
| XMD8-92 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | -2.2 | 10 | uM |
| XMD8-92 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -11.2 | 10 | uM |
| XMD8-92 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | -4.9 | 10 | uM |
| XMD8-92 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -7.0 | 10 | uM |
| XMD8-92 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -15.7 | 10 | uM |
| XMD8-92 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -13.5 | 10 | uM |
| XMD8-92 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 96.0 | 10 | uM |
| XMD8-92 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -8.6 | 10 | uM |
| XMD8-92 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 2.7 | 10 | uM |
| XMD8-92 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -28.7 | 10 | uM |
| XMD8-92 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -12.5 | 10 | uM |
| XMD8-92 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -15.6 | 10 | uM |
| XMD8-92 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -16.3 | 10 | uM |
| XMD8-92 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -18.6 | 10 | uM |
| XMD8-92 | HeLa | ATR | FYIMMCkPK | ATP | -5.7 | 10 | uM |
| XMD8-92 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 40.4 | 10 | uM |
| XMD8-92 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -11.2 | 10 | uM |
| XMD8-92 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -15.5 | 10 | uM |
| XMD8-92 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -20.3 | 10 | uM |
| XMD8-92 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -6.3 | 10 | uM |
| XMD8-92 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | -10.9 | 10 | uM |
| XMD8-92 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | 2.8 | 10 | uM |