XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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  • 1 to 25 of 239 records
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
0.0
10
uM
XMD8-92 PC-3 MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
0.0
10
uM
XMD8-92 HeLa NEK6,NEK7
DIkPANVFITATGVVK
Lys2
0.0
10
uM
XMD8-92 HeLa JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
-0.1
10
uM
XMD8-92 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
0.1
10
uM
XMD8-92 PC-3 SNRK
DLkPENVVFFEK
Lys2
0.3
10
uM
XMD8-92 PC-3 M3K2,MAP3K3
DIkGANILR
Lys2
0.4
10
uM
XMD8-92 HeLa LATS1
ALYATkTLR
Lys1
0.4
10
uM
XMD8-92 PC-3 MST4,YSK1
DIkAANVLLSEQGDVK
Lys2
-0.5
10
uM
XMD8-92 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
0.5
10
uM
XMD8-92 HeLa MLTK
WISQDKEVAVKk
Lys1
-0.8
10
uM
XMD8-92 PC-3 PRP4
CNILHADIkPDNILVNESK
Lys2
0.9
10
uM
XMD8-92 PC-3 CDK5
DLkPQNLLINR
Lys2
-1.0
10
uM
XMD8-92 PC-3 CDK5
NRETHEIVALkR
Lys1
1.0
10
uM
XMD8-92 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
10.0
10
uM
XMD8-92 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
-10.4
10
uM
XMD8-92 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-10.4
10
uM
XMD8-92 PC-3 EPHA2
EVPVAIkTLK
Lys1
-10.5
10
uM
XMD8-92 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
-10.5
10
uM
XMD8-92 PC-3 MAP3K4
DIkGANIFLTSSGLIK
Lys2
10.6
10
uM
XMD8-92 PC-3 JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
10.6
10
uM
XMD8-92 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
10.7
10
uM
XMD8-92 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
10.8
10
uM
XMD8-92 HeLa IRE1
DLkPHNILISMPNAHGK
Lys2
-10.9
10
uM
XMD8-92 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
10.9
10
uM
  • Page 1 of 10
  • 1 to 25 of 239 records