XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | PC-3 | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | 0.0 | 10 | uM |
XMD8-92 | PC-3 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 0.0 | 10 | uM |
XMD8-92 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 0.0 | 10 | uM |
XMD8-92 | HeLa | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | -0.1 | 10 | uM |
XMD8-92 | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 0.1 | 10 | uM |
XMD8-92 | PC-3 | SNRK | DLkPENVVFFEK | Lys2 | 0.3 | 10 | uM |
XMD8-92 | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | 0.4 | 10 | uM |
XMD8-92 | HeLa | LATS1 | ALYATkTLR | Lys1 | 0.4 | 10 | uM |
XMD8-92 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | -0.5 | 10 | uM |
XMD8-92 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 0.5 | 10 | uM |
XMD8-92 | HeLa | MLTK | WISQDKEVAVKk | Lys1 | -0.8 | 10 | uM |
XMD8-92 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | 0.9 | 10 | uM |
XMD8-92 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | -1.0 | 10 | uM |
XMD8-92 | PC-3 | CDK5 | NRETHEIVALkR | Lys1 | 1.0 | 10 | uM |
XMD8-92 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | 10.0 | 10 | uM |
XMD8-92 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | -10.4 | 10 | uM |
XMD8-92 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | -10.4 | 10 | uM |
XMD8-92 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | -10.5 | 10 | uM |
XMD8-92 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | -10.5 | 10 | uM |
XMD8-92 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | 10.6 | 10 | uM |
XMD8-92 | PC-3 | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | 10.6 | 10 | uM |
XMD8-92 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 10.7 | 10 | uM |
XMD8-92 | PC-3 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 10.8 | 10 | uM |
XMD8-92 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | -10.9 | 10 | uM |
XMD8-92 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 10.9 | 10 | uM |