XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -28.7 | 10 | uM |
| XMD8-92 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 40.4 | 10 | uM |
| XMD8-92 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -18.4 | 10 | uM |
| XMD8-92 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -16.3 | 10 | uM |
| XMD8-92 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 11.7 | 10 | uM |
| XMD8-92 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 6.7 | 10 | uM |
| XMD8-92 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 3.9 | 10 | uM |
| XMD8-92 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -15.6 | 10 | uM |
| XMD8-92 | HeLa | ATR | FYIMMCkPK | ATP | -5.7 | 10 | uM |
| XMD8-92 | PC-3 | ATR | FYIMMCkPK | ATP | 6.1 | 10 | uM |
| XMD8-92 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -15.5 | 10 | uM |
| XMD8-92 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -6.3 | 10 | uM |
| XMD8-92 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 2.7 | 10 | uM |
| XMD8-92 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 7.2 | 10 | uM |
| XMD8-92 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 1.6 | 10 | uM |
| XMD8-92 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | -8.1 | 10 | uM |
| XMD8-92 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 2.8 | 10 | uM |
| XMD8-92 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -18.6 | 10 | uM |
| XMD8-92 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 9.2 | 10 | uM |
| XMD8-92 | PC-3 | CDK5 | NRETHEIVALkR | Lys1 | 1.0 | 10 | uM |
| XMD8-92 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -11.2 | 10 | uM |
| XMD8-92 | PC-3 | CDK9 | DMkAANVLITR | Lys2 | -16.1 | 10 | uM |
| XMD8-92 | PC-3 | CHK2 | VAIkIISK | Lys1 | 2.6 | 10 | uM |
| XMD8-92 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | -1.7 | 10 | uM |
| XMD8-92 | PC-3 | CK1d,CK1e | DVkPDNFLMGLGKK | Lys2 | -5.8 | 10 | uM |