HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| HG-6-64-01 | A-375 | TIF1b | VLVNDAQKVTEGQQER | ~NI | 10 | uM | |
| HG-6-64-01 | A-375 | FRAP1 | IQSIAPSLQVITSKQRPR | LIP | ~NI | 10 | uM |
| HG-6-64-01 | A-375 | AGK | ATVFLNPAACKGK | LIP | ~NI | 10 | uM |
| HG-6-64-01 | A-375 | PDK1 | ELATSREYAIKILEKR | K1 | NI | 10 | uM |
| HG-6-64-01 | A-375 | TIF1b | QGSGSSQPMEVQEGYGFGSGDDPYSSAEPHVSGVKR | ND | 10 | uM | |
| HG-6-64-01 | A-375 | SGK3 | DLKPENILLDSVGHVVLTDFGLCK | K2 | ND | 10 | uM |
| HG-6-64-01 | A-375 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | K2 | ND | 10 | uM |
| HG-6-64-01 | A-375 | RPS6KC1 (Domain1) | TEQTFILKGLRK | ND | 10 | uM | |
| HG-6-64-01 | A-375 | MK14 | QELNKTIWEVPER | Other (MAPKAP2/3 active site in p38a complex) | 97.3 | 10 | uM |
| HG-6-64-01 | A-375 | CSK | VSDFGLTKEASSTQDTGKLPVK | ACT | 97.0 | 10 | uM |
| HG-6-64-01 | A-375 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | K2 | 9.7 | 10 | uM |
| HG-6-64-01 | A-375 | ATR | FYIMMCKPK | LIP | 9.7 | 10 | uM |
| HG-6-64-01 | A-375 | LYN | VAVKTLKPGTMSVQAFLEEANLMK | K1 | 96.8 | 10 | uM |
| HG-6-64-01 | A-375 | ABL,ARG | LMTGDTYTAHAGAKFPIK | ACT | 96.2 | 10 | uM |
| HG-6-64-01 | A-375 | AurA,AurB,AurC | GKFGNVYLAR | ATP | 9.6 | 10 | uM |
| HG-6-64-01 | A-375 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | LIP (PI5K) | 9.6 | 10 | uM |
| HG-6-64-01 | A-375 | MAP3K5 | DIKGDNVLINTYSGVLK | K2 | -9.4 | 10 | uM |
| HG-6-64-01 | A-375 | MLTK | WISQDKEVAVKK | K1 | 89.2 | 10 | uM |
| HG-6-64-01 | A-375 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | K2 | 8.8 | 10 | uM |
| HG-6-64-01 | A-375 | MAP3K7,TAK1 | DLKPPNLLLVAGGTVLK | K2 | 86.0 | 10 | uM |
| HG-6-64-01 | A-375 | PKD1,PKD2 | NIVHCDLKPENVLLASADPFPQVK | K2 | 8.4 | 10 | uM |
| HG-6-64-01 | A-375 | EGFR | IPVAIKELR | K1 | -8.3 | 10 | uM |
| HG-6-64-01 | A-375 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | K2 | -7.7 | 10 | uM |
| HG-6-64-01 | A-375 | MLKL | APVAIKVFK | K1 | -7.5 | 10 | uM |
| HG-6-64-01 | A-375 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | ACT | 74.2 | 10 | uM |