PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | IC50 | Conc unit |
---|---|---|---|---|---|---|
PLX-4720 | A-375 | ZC2/TNIK,ZC3/MINK | VIHRDIkGQNVLLTENAEVK | LYS2 | 2.0 | uM |
PLX-4720 | A-375 | ZC2/TNIK | TGQLAAIkVMDVTGDEEEEIKQEINMLKK | LYS1 | 1.2 | uM |
PLX-4720 | A-375 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | LYS2 | 2.0 | uM |
PLX-4720 | A-375 | ZC1/HGK | TGQLAAIkVMDVTEDEEEEIKLEINMLK | LYS1 | 2.2 | uM |
PLX-4720 | A-375 | WNK4 | DLkCDNVFITGPTGSVK | LYS2 | >10 | uM |
PLX-4720 | A-375 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | >10 | uM |
PLX-4720 | A-375 | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | LYS2 | >10 | uM |
PLX-4720 | A-375 | WEE1 | YIHSMSLVHMDIkPSNIFISR | LYS2 | >10 | uM |
PLX-4720 | A-375 | VRK2 | MLDVLEYIHENEYVHGDIkAANLLLGYK | LYS2 | >10 | uM |
PLX-4720 | A-375 | ULK3 | NISHLDLkPQNILLSSLEKPHLK | LYS2 | >10 | uM |
PLX-4720 | A-375 | TLK2 | YVAVkIHQLNK | LYS1 | >10 | uM |
PLX-4720 | A-375 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | LYS2 | >10 | uM |
PLX-4720 | A-375 | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | LYS1 | >10 | uM |
PLX-4720 | A-375 | TAOK2 | DVkAGNILLSEPGLVK | LYS2 | >10 | uM |
PLX-4720 | A-375 | TAO1,TAOK3 | DIkAGNILLTEPGQVK | LYS2 | >10 | uM |
PLX-4720 | A-375 | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | >10 | uM |
PLX-4720 | A-375 | SRC | VAIkTLKPGTMSPEAFLQEAQVMKK | LYS1 | 4.7 | uM |
PLX-4720 | A-375 | SRC | VAIkTLKPGTMSPEAFLQEAQVMK | LYS1 | 3.5 | uM |
PLX-4720 | A-375 | SMG1 | DTVTIHSVGGTITILPTkTKPK | ATP | >10 | uM |
PLX-4720 | A-375 | SLK | DLkAGNILFTLDGDIK | LYS2 | >10 | uM |
PLX-4720 | A-375 | SLK | AQNKETSVLAAAkVIDTK | LYS1 | >10 | uM |
PLX-4720 | A-375 | SLK | IIHRDLkAGNILFTLDGDIK | LYS2 | >10 | uM |
PLX-4720 | A-375 | SGK3 | FYAVkVLQK | LYS1 | 11.0 | uM |
PLX-4720 | A-375 | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | >10 | uM |
PLX-4720 | A-375 | RSK3_domain1 | DLkPENILLDEEGHIKITDFGLSK | LYS2 | >10 | uM |