PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | IC50 | Conc unit |
|---|---|---|---|---|---|---|
| PLX-4720 | A-375 | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | >10 | uM |
| PLX-4720 | A-375 | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | >10 | uM |
| PLX-4720 | A-375 | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Protein Kinase Domain | >10 | uM |
| PLX-4720 | A-375 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | >10 | uM |
| PLX-4720 | A-375 | GCK | DIkGANLLLTLQGDVK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CDK7 | DLkPNNLLLDENGVLK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | GCN2_domain2 | DLkPVNIFLDSDDHVK | LYS2 | 6.4 | uM |
| PLX-4720 | A-375 | Erk5 | DLkPSNLLVNENCELK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | AurA | DIkPENLLLGSAGELK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CDK4 | DLkPENILVTSGGTVK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CDK2 | DLkPQNLLINTEGAIK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CDK9 | DMkAANVLITR | LYS2 | >10 | uM |
| PLX-4720 | A-375 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | BRAF | DLkSNNIFLHEDLTVK | LYS2 | 0.0077 | uM |
| PLX-4720 | A-375 | ARAF | DLkSNNIFLHEGLTVK | LYS2 | 0.022 | uM |
| PLX-4720 | A-375 | DMPK | DIkPDNILLDR | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CHK1 | DIkPENLLLDERDNLK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CK1d,CK1e | DVkPDNFLMGLGKK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CDK5 | NVLHRDLkPQNLLINR | LYS2 | >10 | uM |
| PLX-4720 | A-375 | MK03 | DLkPSNLLINTTCDLK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CDC2 | DLkPQNLLIDDKGTIK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CDK10 | DLkVSNLLMTDK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | CDK11,CDK8 | DLkPANILVMGEGPER | LYS2 | 1.7 | uM |
| PLX-4720 | A-375 | CDK6 | DLkPQNILVTSSGQIK | LYS2 | >10 | uM |
| PLX-4720 | A-375 | KC1A | DIkPDNFLMGIGR | LYS2 | >10 | uM |