QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | MWCL.1 | KC1A | DIKPDNFLMGIGR | Lys2 | -5.104906235 | 1 | uM |
QL-XII-47 | MWCL.1 | CK2a2 | DVKPHNVMIDHQQK | Lys2 | -9.931851645 | 1 | uM |
QL-XII-47 | MWCL.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | -1.027450805 | 1 | uM |
QL-XII-47 | MWCL.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | -20.94285661 | 1 | uM |
QL-XII-47 | MWCL.1 | DNAPK | EHPFLVKGGEDLR | ATP | -17.02227611 | 1 | uM |
QL-XII-47 | MWCL.1 | DNAPK | KGGSWIQEINVAEK | ATP | 14.36767264 | 1 | uM |
QL-XII-47 | MWCL.1 | eEF2K | YIKYNSNSGFVR | ATP | 16.08303464 | 1 | uM |
QL-XII-47 | MWCL.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | ND | 1 | uM |
QL-XII-47 | MWCL.1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | -9.820784106 | 1 | uM |
QL-XII-47 | MWCL.1 | Erk5 | DLKPSNLLVNENCELK | Lys2 | -8.665845057 | 1 | uM |
QL-XII-47 | MWCL.1 | FER | TSVAVKTCKEDLPQELK | Lys1 | 0.548717854 | 1 | uM |
QL-XII-47 | MWCL.1 | FES | LRADNTLVAVKSCR | Lys1 | -6.492258758 | 1 | uM |
QL-XII-47 | MWCL.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | -18.8674785 | 1 | uM |
QL-XII-47 | MWCL.1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | 3.265960592 | 1 | uM |
QL-XII-47 | MWCL.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | -8.174014716 | 1 | uM |
QL-XII-47 | MWCL.1 | GCK | DIKGANLLLTLQGDVK | Lys2 | -4.436115925 | 1 | uM |
QL-XII-47 | MWCL.1 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | -49.83844146 | 1 | uM |
QL-XII-47 | MWCL.1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 5.875370169 | 1 | uM |
QL-XII-47 | MWCL.1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | -5.842092998 | 1 | uM |
QL-XII-47 | MWCL.1 | HPK1 | DIKGANILINDAGEVR | Lys2 | -7.556297789 | 1 | uM |
QL-XII-47 | MWCL.1 | IKKA | DLKPENIVLQDVGGK | Lys2 | -1.846234471 | 1 | uM |
QL-XII-47 | MWCL.1 | IKKB | DLKPENIVLQQGEQR | Lys2 | 0.88441842 | 1 | uM |
QL-XII-47 | MWCL.1 | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | 0.982360401 | 1 | uM |
QL-XII-47 | MWCL.1 | ILK | WQGNDIVVKVLK | Lys1 | 3.920530194 | 1 | uM |
QL-XII-47 | MWCL.1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 29.07160077 | 1 | uM |