QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 BCWM.1 NEK9
DIKTLNIFLTK
Lys2
-8.692345813
1
uM
QL-XII-47 BCWM.1 OSR1
DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR
Lys2
-2.037568348
1
uM
QL-XII-47 BCWM.1 p38a
DLKPSNLAVNEDCELK
Lys2
-8.718461078
1
uM
QL-XII-47 BCWM.1 MK14
QELNKTIWEVPER
Other
-2.012618075
1
uM
QL-XII-47 BCWM.1 MK11
QELNKTVWEVPQR
Other
9.053676509
1
uM
QL-XII-47 BCWM.1 p38d,p38g
DLKPGNLAVNEDCELK
Lys2
1.738509549
1
uM
QL-XII-47 BCWM.1 KS6B1
DLKPENIMLNHQGHVK
Lys2
23.62820654
1
uM
QL-XII-47 BCWM.1 KS6B2
DLKPENIMLSSQGHIK
Lys2
6.904041963
1
uM
QL-XII-47 BCWM.1 PAN3
VMDPTKILITGK
ATP
34.20265652
1
uM
QL-XII-47 BCWM.1 PCTAIRE2,PCTAIRE3
SKLTENLVALKEIR
Lys1
-7.31403483
1
uM
QL-XII-47 BCWM.1 PDK1
EYAIKILEK
Lys1
-13.88134428
1
uM
QL-XII-47 BCWM.1 PEK
DLKPSNIFFTMDDVVK
Lys2
11.19892963
1
uM
QL-XII-47 BCWM.1 CDK14
LVALKVIR
Lys1
20.63298661
1
uM
QL-XII-47 BCWM.1 PHKg2
ATGHEFAVKIMEVTAER
Lys1
22.98766626
1
uM
QL-XII-47 BCWM.1 PI4KA,PI4KAP2
SGTPMQSAAKAPYLAK
ATP
3.960959449
1
uM
QL-XII-47 BCWM.1 PI4KB
VPHTQAVVLNSKDK
ATP
7.838958764
1
uM
QL-XII-47 BCWM.1 PIK3C2B
VIFKCGDDLRQDMLTLQMIR
ATP
3.467990236
1
uM
QL-XII-47 BCWM.1 PIK3C3
TEDGGKYPVIFKHGDDLR
ATP
-15.19310639
1
uM
QL-XII-47 BCWM.1 PIK3CB
VFGEDSVGVIFKNGDDLRQDMLTLQMLR
ATP
22.61758294
1
uM
QL-XII-47 BCWM.1 PIK3CD
VNWLAHNVSKDNRQ
ATP
-2.373774845
1
uM
QL-XII-47 BCWM.1 PIK3CG
KKPLWLEFK
ATP
-49.28259781
1
uM
QL-XII-47 BCWM.1 PIP4K2A
AKELPTLKDNDFINEGQK
ATP
-5.721584145
1
uM
QL-XII-47 BCWM.1 PI42C
TLVIKEVSSEDIADMHSNLSNYHQYIVK
ATP
4.443788957
1
uM
QL-XII-47 BCWM.1 FYV1
GGKSGAAFYATEDDRFILK
ATP
9.038475869
1
uM
QL-XII-47 BCWM.1 PITSLRE
DLKTSNLLLSHAGILK
Lys2
-21.97942299
1
uM