QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 BCWM.1 MARK3
EVAIKIIDKTQLNPTSLQK
Lys1
-9.506780432
1
uM
QL-XII-47 BCWM.1 MARK3,MARK4
EVAIKIIDK
Lys1
-5.245158983
1
uM
QL-XII-47 BCWM.1 MAST1,MAST2
DLKPDNLLITSMGHIK
Lys2
-49.97672913
1
uM
QL-XII-47 BCWM.1 MAST3
DLKPDNLLITSLGHIK
Lys2
-14.29780438
1
uM
QL-XII-47 BCWM.1 MASTL
GAFGKVYLGQK
ATP Loop
-0.133762637
1
uM
QL-XII-47 BCWM.1 MASTL
LYAVKVVK
Lys1
3.164579615
1
uM
QL-XII-47 BCWM.1 MLK3
DLKSNNILLLQPIESDDMEHK
Lys2
6.517393593
1
uM
QL-XII-47 BCWM.1 MLK4
DLKSSNILLLEK
Lys2
25.06956525
1
uM
QL-XII-47 BCWM.1 MLKL
APVAIKVFK
Lys1
-8.7509279
1
uM
QL-XII-47 BCWM.1 MSK1_domain1
DIKLENILLDSNGHVVLTDFGLSK
Lys2
-19.81407645
1
uM
QL-XII-47 BCWM.1 MSK2 domain1
DLKLENVLLDSEGHIVLTDFGLSK
Lys2
-46.59383779
1
uM
QL-XII-47 BCWM.1 MST1
ETGQIVAIKQVPVESDLQEIIK
Lys1
12.32676416
1
uM
QL-XII-47 BCWM.1 MST2
ESGQVVAIKQVPVESDLQEIIK
Lys1
9.022179848
1
uM
QL-XII-47 BCWM.1 MST3
DIKAANVLLSEHGEVK
Lys2
-7.32686656
1
uM
QL-XII-47 BCWM.1 MST4
TQQVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSSYVTK
Lys1
4.712110007
1
uM
QL-XII-47 BCWM.1 MST4,YSK1
DIKAANVLLSEQGDVK
Lys2
-12.31136342
1
uM
QL-XII-47 BCWM.1 MYO3A,MYO3B
DVKGNNILLTTEGGVK
Lys2
22.46529411
1
uM
QL-XII-47 BCWM.1 NDR1
DIKPDNLLLDSK
Lys2
8.69546525
1
uM
QL-XII-47 BCWM.1 NDR2
DIKPDNLLLDAK
Lys2
21.26831557
1
uM
QL-XII-47 BCWM.1 NEK1
DIKSQNIFLTK
Lys2
13.37762142
1
uM
QL-XII-47 BCWM.1 NEK3
SKNIFLTQNGK
Activation Loop
-10.13654488
1
uM
QL-XII-47 BCWM.1 NEK4
DLKTQNVFLTR
Lys2
8.402917665
1
uM
QL-XII-47 BCWM.1 NEK6,NEK7
DIKPANVFITATGVVK
Lys2
-20.01162346
1
uM
QL-XII-47 BCWM.1 NEK7
AACLLDGVPVALKK
Lys1
-3.686949487
1
uM
QL-XII-47 BCWM.1 NEK8
DLKTQNILLDK
Lys2
9.444227339
1
uM