QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | BCWM.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | -9.506780432 | 1 | uM |
QL-XII-47 | BCWM.1 | MARK3,MARK4 | EVAIKIIDK | Lys1 | -5.245158983 | 1 | uM |
QL-XII-47 | BCWM.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | -49.97672913 | 1 | uM |
QL-XII-47 | BCWM.1 | MAST3 | DLKPDNLLITSLGHIK | Lys2 | -14.29780438 | 1 | uM |
QL-XII-47 | BCWM.1 | MASTL | GAFGKVYLGQK | ATP Loop | -0.133762637 | 1 | uM |
QL-XII-47 | BCWM.1 | MASTL | LYAVKVVK | Lys1 | 3.164579615 | 1 | uM |
QL-XII-47 | BCWM.1 | MLK3 | DLKSNNILLLQPIESDDMEHK | Lys2 | 6.517393593 | 1 | uM |
QL-XII-47 | BCWM.1 | MLK4 | DLKSSNILLLEK | Lys2 | 25.06956525 | 1 | uM |
QL-XII-47 | BCWM.1 | MLKL | APVAIKVFK | Lys1 | -8.7509279 | 1 | uM |
QL-XII-47 | BCWM.1 | MSK1_domain1 | DIKLENILLDSNGHVVLTDFGLSK | Lys2 | -19.81407645 | 1 | uM |
QL-XII-47 | BCWM.1 | MSK2 domain1 | DLKLENVLLDSEGHIVLTDFGLSK | Lys2 | -46.59383779 | 1 | uM |
QL-XII-47 | BCWM.1 | MST1 | ETGQIVAIKQVPVESDLQEIIK | Lys1 | 12.32676416 | 1 | uM |
QL-XII-47 | BCWM.1 | MST2 | ESGQVVAIKQVPVESDLQEIIK | Lys1 | 9.022179848 | 1 | uM |
QL-XII-47 | BCWM.1 | MST3 | DIKAANVLLSEHGEVK | Lys2 | -7.32686656 | 1 | uM |
QL-XII-47 | BCWM.1 | MST4 | TQQVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSSYVTK | Lys1 | 4.712110007 | 1 | uM |
QL-XII-47 | BCWM.1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | -12.31136342 | 1 | uM |
QL-XII-47 | BCWM.1 | MYO3A,MYO3B | DVKGNNILLTTEGGVK | Lys2 | 22.46529411 | 1 | uM |
QL-XII-47 | BCWM.1 | NDR1 | DIKPDNLLLDSK | Lys2 | 8.69546525 | 1 | uM |
QL-XII-47 | BCWM.1 | NDR2 | DIKPDNLLLDAK | Lys2 | 21.26831557 | 1 | uM |
QL-XII-47 | BCWM.1 | NEK1 | DIKSQNIFLTK | Lys2 | 13.37762142 | 1 | uM |
QL-XII-47 | BCWM.1 | NEK3 | SKNIFLTQNGK | Activation Loop | -10.13654488 | 1 | uM |
QL-XII-47 | BCWM.1 | NEK4 | DLKTQNVFLTR | Lys2 | 8.402917665 | 1 | uM |
QL-XII-47 | BCWM.1 | NEK6,NEK7 | DIKPANVFITATGVVK | Lys2 | -20.01162346 | 1 | uM |
QL-XII-47 | BCWM.1 | NEK7 | AACLLDGVPVALKK | Lys1 | -3.686949487 | 1 | uM |
QL-XII-47 | BCWM.1 | NEK8 | DLKTQNILLDK | Lys2 | 9.444227339 | 1 | uM |