QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | BCWM.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | -18.81736377 | 1 | uM |
| QL-XII-47 | BCWM.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | -55.6912494 | 1 | uM |
| QL-XII-47 | BCWM.1 | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | -18.18174987 | 1 | uM |
| QL-XII-47 | BCWM.1 | KHS1 | NVHTGELAAVKIIK | Lys1 | -5.41406842 | 1 | uM |
| QL-XII-47 | BCWM.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | -18.43797163 | 1 | uM |
| QL-XII-47 | BCWM.1 | LATS1 | ALYATKTLR | Lys1 | 4.639137919 | 1 | uM |
| QL-XII-47 | BCWM.1 | LATS2 | DIKPDNILIDLDGHIK | Lys2 | -6.394868054 | 1 | uM |
| QL-XII-47 | BCWM.1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | -1.155961788 | 1 | uM |
| QL-XII-47 | BCWM.1 | LOK | DLKAGNVLMTLEGDIR | Lys2 | 27.92541625 | 1 | uM |
| QL-XII-47 | BCWM.1 | LRRK2 | DLKPHNVLLFTLYPNAAIIAK | Lys2 | -8.514705323 | 1 | uM |
| QL-XII-47 | BCWM.1 | LYN | VAVKTLKPGTMSVQAFLEEANLMK | Lys1 | 5.664881312 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP2K1 | IMHRDVKPSNILVNSR | Lys2 | 8.135028611 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | 1.156231522 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP2K3 | DVKPSNVLINK | Lys2 | -1.51563755 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP2K4 | DIKPSNILLDR | Lys2 | -0.827779834 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP2K5 | DVKPSNMLVNTR | Lys2 | 19.59807956 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP2K6 | DVKPSNVLINALGQVK | Lys2 | -2.952147998 | 1 | uM |
| QL-XII-47 | BCWM.1 | MP2K7 | DVKPSNILLDER | Lys2 | -16.63595781 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | -4.774099061 | 1 | uM |
| QL-XII-47 | BCWM.1 | M3K2 | ELAVKQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -1.41395978 | 1 | uM |
| QL-XII-47 | BCWM.1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | 14.75543663 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP3K3 | ELASKQVQFDPDSPETSKEVSALECEIQLLK | Lys1 | 1.847720029 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | 22.67873912 | 1 | uM |
| QL-XII-47 | BCWM.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | -4.886038638 | 1 | uM |
| QL-XII-47 | BCWM.1 | MARK2,MARK3 | DLKAENLLLDADMNIK | Lys2 | 13.21947164 | 1 | uM |