QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | MWCL.1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 10.33171657 | 1 | uM |
| QL-XII-47 | MWCL.1 | IRE1 | DLKPHNILISMPNAHGK | Lys2 | -7.659764425 | 1 | uM |
| QL-XII-47 | MWCL.1 | ITPK1 | ESIFFNSHNVSKPESSSVLTELDKIEGVFERPSDEVIR | ATP | 22.80886811 | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK1 | QLASALSYLEDKDLVHGNVCTKNLLLAR | Other | 33.14187264 | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | -9.341503001 | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | -87.4730226 | 1 | uM |
| QL-XII-47 | MWCL.1 | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | 2.513675969 | 1 | uM |
| QL-XII-47 | MWCL.1 | KHS1 | NVHTGELAAVKIIK | Lys1 | 10.44210585 | 1 | uM |
| QL-XII-47 | MWCL.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | -17.85533882 | 1 | uM |
| QL-XII-47 | MWCL.1 | LATS1 | ALYATKTLR | Lys1 | 13.55275871 | 1 | uM |
| QL-XII-47 | MWCL.1 | LATS2 | DIKPDNILIDLDGHIK | Lys2 | 13.48092935 | 1 | uM |
| QL-XII-47 | MWCL.1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 5.905585783 | 1 | uM |
| QL-XII-47 | MWCL.1 | LOK | DLKAGNVLMTLEGDIR | Lys2 | -3.152905014 | 1 | uM |
| QL-XII-47 | MWCL.1 | LRRK2 | DLKPHNVLLFTLYPNAAIIAK | Lys2 | 7.098641111 | 1 | uM |
| QL-XII-47 | MWCL.1 | LYN | VAVKTLKPGTMSVQAFLEEANLMK | Lys1 | 2.528406343 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP2K1 | IMHRDVKPSNILVNSR | Lys2 | -10.45585154 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | 2.14775294 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP2K3 | DVKPSNVLINK | Lys2 | -11.1285874 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP2K4 | DIKPSNILLDR | Lys2 | -4.661208852 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP2K5 | DVKPSNMLVNTR | Lys2 | -4.198608382 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP2K6 | DVKPSNVLINALGQVK | Lys2 | 5.39398113 | 1 | uM |
| QL-XII-47 | MWCL.1 | MP2K7 | DVKPSNILLDER | Lys2 | -45.5174114 | 1 | uM |
| QL-XII-47 | MWCL.1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | 9.175244255 | 1 | uM |
| QL-XII-47 | MWCL.1 | M3K2 | ELAVKQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -0.459368027 | 1 | uM |
| QL-XII-47 | MWCL.1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | 17.59521009 | 1 | uM |