NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NPK76-II-72-1 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | -25.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | 69.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -19.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | 12.6 | 10 | uM |
| NPK76-II-72-1 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -16.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -4.9 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | -12.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | TLK1 | YAAVkIHQLNK | Lys1 | -9.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | -4.3 | 10 | uM |
| NPK76-II-72-1 | PC-3 | ILK | WQGNDIVVkVLK | Lys1 | -18.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | -11.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | MLTK | WISQDKEVAVKk | Lys1 | -31.1 | 10 | uM |
| NPK76-II-72-1 | PC-3 | M3K2 | VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | 5.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -11.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -5.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 0.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -7.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | PAN3 | VMDPTkILITGK | -19.2 | 10 | uM | |
| NPK76-II-72-1 | HeLa | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | -207.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | -9.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | -11.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -2.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 16.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -0.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | -6.7 | 10 | uM |