NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NPK76-II-72-1 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | -4.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | -44.1 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | 4.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 16.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | -58.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | SYK | ISDFGLSkALR | Activation Loop | -12.9 | 10 | uM |
| NPK76-II-72-1 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -5.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | -16.7 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | -79.9 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | -5.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | RSK2_domain1 | LTDFGLSkESIDHEKK | Activation Loop | -7.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | -0.9 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | -13.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | RSK1 domain1 | LTDFGLSkEAIDHEK | Activation Loop | -26.1 | 10 | uM |
| NPK76-II-72-1 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -31.1 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -11.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | 69.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -4.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | -25.1 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -2.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 10.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -20.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -0.3 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 0.4 | 10 | uM |
| NPK76-II-72-1 | HeLa | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 38.8 | 10 | uM |