NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
NPK76-II-72-1 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -31.1 | 10 | uM |
NPK76-II-72-1 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | -1.0 | 10 | uM |
NPK76-II-72-1 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -1.8 | 10 | uM |
NPK76-II-72-1 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | -30.6 | 10 | uM |
NPK76-II-72-1 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -14.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 20.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 11.3 | 10 | uM |
NPK76-II-72-1 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | -35.6 | 10 | uM |
NPK76-II-72-1 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -2.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | ATR | FYIMMCkPK | ATP | 7.4 | 10 | uM |
NPK76-II-72-1 | HeLa | ATR | FYIMMCkPK | ATP | -80.8 | 10 | uM |
NPK76-II-72-1 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | 9.7 | 10 | uM |
NPK76-II-72-1 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | -6.5 | 10 | uM |
NPK76-II-72-1 | HeLa | BTK | GQYDVAIkMIK | Lys1 | -27.4 | 10 | uM |
NPK76-II-72-1 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | 10.8 | 10 | uM |
NPK76-II-72-1 | HeLa | CAMK1D | LFAVkCIPK | Lys1 | 17.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 65.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 64.5 | 10 | uM |
NPK76-II-72-1 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 63.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | -33.4 | 10 | uM |
NPK76-II-72-1 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | -14.6 | 10 | uM |
NPK76-II-72-1 | PC-3 | CDK14 | LVALkVIR | Lys1 | 3.0 | 10 | uM |
NPK76-II-72-1 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | -9.4 | 10 | uM |
NPK76-II-72-1 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 0.5 | 10 | uM |
NPK76-II-72-1 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -10.5 | 10 | uM |