NPK76-II-72-1 KiNativ -- single dose experiment - Dataset (ID:20106)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NPK76-II-72-1 | PC-3 | LOK | DLkAGNVLMTLEGDIR | Lys2 | -0.2 | 10 | uM |
| NPK76-II-72-1 | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 0.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -0.3 | 10 | uM |
| NPK76-II-72-1 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -0.3 | 10 | uM |
| NPK76-II-72-1 | PC-3 | KHS1 | NVHTGELAAVkIIK | Lys1 | 0.3 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 0.4 | 10 | uM |
| NPK76-II-72-1 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | -0.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 0.5 | 10 | uM |
| NPK76-II-72-1 | HeLa | PKR | DLkPSNIFLVDTK | Lys2 | 0.6 | 10 | uM |
| NPK76-II-72-1 | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 0.6 | 10 | uM |
| NPK76-II-72-1 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | -0.9 | 10 | uM |
| NPK76-II-72-1 | HeLa | MSK1_domain1 | DIkLENILLDSNGHVVLTDFGLSK | Lys2 | -0.9 | 10 | uM |
| NPK76-II-72-1 | PC-3 | RON | IQCAIkSLSR | Lys1 | -1.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | -1.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -10.1 | 10 | uM |
| NPK76-II-72-1 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -10.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 10.3 | 10 | uM |
| NPK76-II-72-1 | PC-3 | M4K3 | NVNTGELAAIkVIK | Lys1 | 10.4 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -10.5 | 10 | uM |
| NPK76-II-72-1 | PC-3 | EGFR | IPVAIkELR | Lys1 | 10.7 | 10 | uM |
| NPK76-II-72-1 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | 10.8 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -11.0 | 10 | uM |
| NPK76-II-72-1 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | 11.0 | 10 | uM |
| NPK76-II-72-1 | HeLa | PKD2 | DVAVkVIDK | Lys1 | -11.2 | 10 | uM |
| NPK76-II-72-1 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | -11.3 | 10 | uM |