JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JWE-035 | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | 0.0 | 10 | uM |
| JWE-035 | HeLa | SYK | ISDFGLSkALR | Activation Loop | -0.1 | 10 | uM |
| JWE-035 | PC-3 | MAP2K4 | DIkPSNILLDR | Lys2 | -0.3 | 10 | uM |
| JWE-035 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -0.3 | 10 | uM |
| JWE-035 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | 0.3 | 10 | uM |
| JWE-035 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | -0.4 | 10 | uM |
| JWE-035 | HeLa | SMG1 | DTVTIHSVGGTITILPTkTKPK | ATP | -0.6 | 10 | uM |
| JWE-035 | HeLa | DGKA | IDPVPNTHPLLVFVNPkSGGK | ATP | -0.7 | 10 | uM |
| JWE-035 | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | -0.7 | 10 | uM |
| JWE-035 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 0.7 | 10 | uM |
| JWE-035 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | 0.8 | 10 | uM |
| JWE-035 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -0.9 | 10 | uM |
| JWE-035 | HeLa | PKN1 | GHFGkVLLSEFRPSGELFAIK | Lys1 | -10.0 | 10 | uM |
| JWE-035 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | -10.2 | 10 | uM |
| JWE-035 | HeLa | PIK3CG | KkPLWLEFK | ATP | 10.2 | 10 | uM |
| JWE-035 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | 10.2 | 10 | uM |
| JWE-035 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -10.4 | 10 | uM |
| JWE-035 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | 10.5 | 10 | uM |
| JWE-035 | PC-3 | NEK8 | DLkTQNILLDK | Lys2 | 10.6 | 10 | uM |
| JWE-035 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | 10.7 | 10 | uM |
| JWE-035 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | 10.9 | 10 | uM |
| JWE-035 | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | -1.1 | 10 | uM |
| JWE-035 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -1.1 | 10 | uM |
| JWE-035 | HeLa | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | 1.1 | 10 | uM |
| JWE-035 | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | 11.5 | 10 | uM |