JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
JWE-035 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -9.9 | 10 | uM |
JWE-035 | PC-3 | SRPK1 | IIHTDIkPENILLSVNEQYIR | Lys2 | 9.8 | 10 | uM |
JWE-035 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | 9.7 | 10 | uM |
JWE-035 | HeLa | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 9.6 | 10 | uM |
JWE-035 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 95.4 | 10 | uM |
JWE-035 | HeLa | KPCI | IYAMkVVK | Lys1 | 9.4 | 10 | uM |
JWE-035 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | 9.4 | 10 | uM |
JWE-035 | HeLa | RSK1 domain1 | LTDFGLSkEAIDHEK | Activation Loop | -9.4 | 10 | uM |
JWE-035 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | 93.2 | 10 | uM |
JWE-035 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 9.2 | 10 | uM |
JWE-035 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 91.1 | 10 | uM |
JWE-035 | HeLa | LATS1 | ALYATkTLR | Lys1 | -8.8 | 10 | uM |
JWE-035 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -8.8 | 10 | uM |
JWE-035 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | 8.5 | 10 | uM |
JWE-035 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | 8.4 | 10 | uM |
JWE-035 | PC-3 | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | 8.4 | 10 | uM |
JWE-035 | PC-3 | PKR | DLkPSNIFLVDTK | Lys2 | 8.4 | 10 | uM |
JWE-035 | HeLa | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 83.0 | 10 | uM |
JWE-035 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | 8.2 | 10 | uM |
JWE-035 | HeLa | ATR | FYIMMCkPK | ATP | 8.1 | 10 | uM |
JWE-035 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | -8.1 | 10 | uM |
JWE-035 | HeLa | AurB | SHFIVALkVLFK | Lys1 | 80.4 | 10 | uM |
JWE-035 | PC-3 | MAP2K3 | DVkPSNVLINK | Lys2 | 7.9 | 10 | uM |
JWE-035 | HeLa | MK14 | QELNkTIWEVPER | Other | 7.9 | 10 | uM |
JWE-035 | HeLa | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 7.9 | 10 | uM |