JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JWE-035 | PC-3 | IRAK1 | AIQFLHQDSPSLIHGDIkSSNVLLDER | Lys2 | 19.9 | 10 | uM |
| JWE-035 | HeLa | LATS1 | ALYATkTLR | Lys1 | -8.8 | 10 | uM |
| JWE-035 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | 2.4 | 10 | uM |
| JWE-035 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -18.2 | 10 | uM |
| JWE-035 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 34.0 | 10 | uM |
| JWE-035 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -0.9 | 10 | uM |
| JWE-035 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | 17.5 | 10 | uM |
| JWE-035 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | 25.8 | 10 | uM |
| JWE-035 | PC-3 | MST1,MST2 | DIkAGNILLNTEGHAK | Lys2 | -33.0 | 10 | uM |
| JWE-035 | PC-3 | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | 31.5 | 10 | uM |
| JWE-035 | HeLa | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | -2.0 | 10 | uM |
| JWE-035 | HeLa | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | 1.1 | 10 | uM |
| JWE-035 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | 21.0 | 10 | uM |
| JWE-035 | HeLa | M3K2,MAP3K3 | DIkGANILR | Lys2 | -3.7 | 10 | uM |
| JWE-035 | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | 25.3 | 10 | uM |
| JWE-035 | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | -1.1 | 10 | uM |
| JWE-035 | HeLa | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 3.8 | 10 | uM |
| JWE-035 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 3.1 | 10 | uM |
| JWE-035 | HeLa | MSK1_domain1 | DIkLENILLDSNGHVVLTDFGLSK | Lys2 | 2.8 | 10 | uM |
| JWE-035 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -2.8 | 10 | uM |
| JWE-035 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 6.5 | 10 | uM |
| JWE-035 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | -0.4 | 10 | uM |
| JWE-035 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -5.1 | 10 | uM |
| JWE-035 | PC-3 | MRCKb | DIkPDNVLLDVNGHIR | Lys2 | 4.7 | 10 | uM |
| JWE-035 | HeLa | CHK1 | DIkPENLLLDER | Lys2 | -6.0 | 10 | uM |