JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JWE-035 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | 10.2 | 10 | uM |
| JWE-035 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 55.4 | 10 | uM |
| JWE-035 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 29.7 | 10 | uM |
| JWE-035 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | 14.6 | 10 | uM |
| JWE-035 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -1.7 | 10 | uM |
| JWE-035 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | 0.3 | 10 | uM |
| JWE-035 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 3.2 | 10 | uM |
| JWE-035 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -5.1 | 10 | uM |
| JWE-035 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -9.9 | 10 | uM |
| JWE-035 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 95.4 | 10 | uM |
| JWE-035 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -5.7 | 10 | uM |
| JWE-035 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 19.9 | 10 | uM |
| JWE-035 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 91.1 | 10 | uM |
| JWE-035 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | 10.5 | 10 | uM |
| JWE-035 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | 6.2 | 10 | uM |
| JWE-035 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 63.0 | 10 | uM |
| JWE-035 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 6.7 | 10 | uM |
| JWE-035 | HeLa | ATR | FYIMMCkPK | ATP | 8.1 | 10 | uM |
| JWE-035 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 30.9 | 10 | uM |
| JWE-035 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | 54.2 | 10 | uM |
| JWE-035 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 4.5 | 10 | uM |
| JWE-035 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | 4.2 | 10 | uM |
| JWE-035 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | 0.8 | 10 | uM |
| JWE-035 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | 6.6 | 10 | uM |
| JWE-035 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -6.1 | 10 | uM |