XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

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  • 1 to 25 of 241 records
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
41.9
10
uM
XMD16-144 HeLa SYK
ISDFGLSkALR
Activation Loop
14.5
10
uM
XMD16-144 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
0.2
10
uM
XMD16-144 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
-7.5
10
uM
XMD16-144 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
4.5
10
uM
XMD16-144 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-4.7
10
uM
XMD16-144 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
13.9
10
uM
XMD16-144 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
26.1
10
uM
XMD16-144 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
-2.5
10
uM
XMD16-144 PC-3 NEK9
LGDYGLAkK
Activation Loop
8.6
10
uM
XMD16-144 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
11.1
10
uM
XMD16-144 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
43.9
10
uM
XMD16-144 HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
-48.5
10
uM
XMD16-144 PC-3 MET
DMYDKEYYSVHNkTGAK
Activation Loop
57.2
10
uM
XMD16-144 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
83.8
10
uM
XMD16-144 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-2.0
10
uM
XMD16-144 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
10
uM
XMD16-144 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
19.4
10
uM
XMD16-144 HeLa JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
-1.6
10
uM
XMD16-144 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
66.9
10
uM
XMD16-144 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
4.4
10
uM
XMD16-144 HeLa NEK9
LGDYGLAkK
Activation Loop
1.5
10
uM
XMD16-144 HeLa RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
24.3
10
uM
XMD16-144 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
27.3
10
uM
XMD16-144 HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
36.3
10
uM
  • Page 1 of 10
  • 1 to 25 of 241 records