XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD16-144 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | 41.9 | 10 | uM |
XMD16-144 | HeLa | SYK | ISDFGLSkALR | Activation Loop | 14.5 | 10 | uM |
XMD16-144 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | 0.2 | 10 | uM |
XMD16-144 | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | -7.5 | 10 | uM |
XMD16-144 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | 4.5 | 10 | uM |
XMD16-144 | HeLa | RSK1 domain1 | LTDFGLSkEAIDHEK | Activation Loop | -4.7 | 10 | uM |
XMD16-144 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 13.9 | 10 | uM |
XMD16-144 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 26.1 | 10 | uM |
XMD16-144 | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | -2.5 | 10 | uM |
XMD16-144 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 8.6 | 10 | uM |
XMD16-144 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 11.1 | 10 | uM |
XMD16-144 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 43.9 | 10 | uM |
XMD16-144 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | -48.5 | 10 | uM |
XMD16-144 | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | 57.2 | 10 | uM |
XMD16-144 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 83.8 | 10 | uM |
XMD16-144 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -2.0 | 10 | uM |
XMD16-144 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | 10 | uM | |
XMD16-144 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | 19.4 | 10 | uM |
XMD16-144 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | -1.6 | 10 | uM |
XMD16-144 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 66.9 | 10 | uM |
XMD16-144 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 4.4 | 10 | uM |
XMD16-144 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | 1.5 | 10 | uM |
XMD16-144 | HeLa | RSK2_domain1 | LTDFGLSkESIDHEKK | Activation Loop | 24.3 | 10 | uM |
XMD16-144 | HeLa | TEC | YVLDDQYTSSSGAkFPVK | Activation Loop | 27.3 | 10 | uM |
XMD16-144 | HeLa | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | 36.3 | 10 | uM |