XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD16-144 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | 0.0 | 10 | uM |
| XMD16-144 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | 0.0 | 10 | uM |
| XMD16-144 | PC-3 | KHS1 | NVHTGELAAVkIIK | Lys1 | -0.1 | 10 | uM |
| XMD16-144 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | 0.2 | 10 | uM |
| XMD16-144 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | 0.2 | 10 | uM |
| XMD16-144 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -0.7 | 10 | uM |
| XMD16-144 | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | -0.9 | 10 | uM |
| XMD16-144 | HeLa | LATS1 | ALYATkTLR | Lys1 | -1.0 | 10 | uM |
| XMD16-144 | HeLa | ILK | WQGIVVkVLK | Lys1 | 1.0 | 10 | uM |
| XMD16-144 | PC-3 | CLK2 | LTHTDLkPENILFVNSDYELTYNLEK | Lys2 | 10.0 | 10 | uM |
| XMD16-144 | PC-3 | TLK1 | YAAVkIHQLNK | Lys1 | -10.1 | 10 | uM |
| XMD16-144 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | 10.2 | 10 | uM |
| XMD16-144 | PC-3 | MAP2K6 | DVkPSNVLINALGQVK | Lys2 | -10.3 | 10 | uM |
| XMD16-144 | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | -10.3 | 10 | uM |
| XMD16-144 | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 10.8 | 10 | uM |
| XMD16-144 | HeLa | CAMK1D | LFAVkCIPK | Lys1 | 10.8 | 10 | uM |
| XMD16-144 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -11.0 | 10 | uM |
| XMD16-144 | HeLa | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 11.0 | 10 | uM |
| XMD16-144 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 11.1 | 10 | uM |
| XMD16-144 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | 11.3 | 10 | uM |
| XMD16-144 | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | 11.4 | 10 | uM |
| XMD16-144 | PC-3 | PRPK | FLSGLELVkQGAEAR | ATP Loop | -11.8 | 10 | uM |
| XMD16-144 | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | 11.8 | 10 | uM |
| XMD16-144 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -11.9 | 10 | uM |
| XMD16-144 | PC-3 | RON | IQCAIkSLSR | Lys1 | -1.2 | 10 | uM |