XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD16-144 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 83.8 | 10 | uM |
| XMD16-144 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 79.4 | 10 | uM |
| XMD16-144 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -17.8 | 10 | uM |
| XMD16-144 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 91.3 | 10 | uM |
| XMD16-144 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 93.6 | 10 | uM |
| XMD16-144 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 90.9 | 10 | uM |
| XMD16-144 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 91.3 | 10 | uM |
| XMD16-144 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | -30.6 | 10 | uM |
| XMD16-144 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | -20.3 | 10 | uM |
| XMD16-144 | PC-3 | ATR | FYIMMCkPK | ATP | -16.0 | 10 | uM |
| XMD16-144 | HeLa | ATR | FYIMMCkPK | ATP | -22.3 | 10 | uM |
| XMD16-144 | HeLa | AurB | SHFIVALkVLFK | Lys1 | 97.3 | 10 | uM |
| XMD16-144 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | 1.7 | 10 | uM |
| XMD16-144 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 7.5 | 10 | uM |
| XMD16-144 | HeLa | BTK | GQYDVAIkMIK | Lys1 | -35.4 | 10 | uM |
| XMD16-144 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | 4.2 | 10 | uM |
| XMD16-144 | HeLa | CAMK1D | LFAVkCIPK | Lys1 | 10.8 | 10 | uM |
| XMD16-144 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 42.2 | 10 | uM |
| XMD16-144 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 47.3 | 10 | uM |
| XMD16-144 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 39.3 | 10 | uM |
| XMD16-144 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 26.8 | 10 | uM |
| XMD16-144 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | 49.2 | 10 | uM |
| XMD16-144 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 16.6 | 10 | uM |
| XMD16-144 | PC-3 | CDK14 | LVALkVIR | Lys1 | -2.9 | 10 | uM |
| XMD16-144 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | 4.2 | 10 | uM |